SCHEMBL6024164

SCHEMBL6024164

CCCCC[C@H](CNC(=O)OCc1ccccc1)C(=O)NN(CCCC)C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.49
MAPT P10636 1/20 0.44
CTSL P07711 1/20 0.43
CTSS P25774 1/20 0.43
SIRT2 Q8IXJ6 6/20 0.43
SIRT1 Q96EB6 3/20 0.42
SIRT3 Q9NTG7 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1596256 0.84 SYK (0.40) SYKMAPTCTSLCTSS
SCHEMBL3722611 0.84 SYK (0.50) SYK
SCHEMBL13434967 0.81 SIRT2 (0.53) SYKCTSLCTSSSIRT2SIRT1
SCHEMBL3902571 0.81 SIRT2 (0.53) SYKCTSLCTSSSIRT2SIRT1
SCHEMBL133032 0.81 SIRT2 (0.53) SYKCTSLCTSSSIRT2SIRT1
SCHEMBL1596691 0.81 CTSL (0.52) SYKCTSLCTSSSIRT2SIRT1
SCHEMBL8054994 0.80 SIRT2 (0.55) SYKCTSLCTSSSIRT2SIRT1
SCHEMBL6024571 0.80 L3MBTL1 (0.41)
SCHEMBL25002520 0.78 SYK (0.53) SYKMAPTCTSL
SCHEMBL3319289 0.78 CTSL (0.56) SYKMAPTCTSLCTSSSIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1363873-B1 PEPTIDE DEFORMYLASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2016-04-20 EP disclosed
US-7019003-B2 Peptide deformylase inhibitors SMITHKLINE BEECHAM CORPORATION (US) 2006-03-28 US disclosed
EP-1363873-A4 PEPTIDE DEFORMYLASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2006-01-04 EP disclosed
US-20040087585-A1 Peptide deformylase inhibitors GLAXOSMITHKLINE LLC 2004-05-06 US disclosed
EP-1363873-A2 PEPTIDE DEFORMYLASE INHIBITORS SmithKline Beecham Corporation (US) 2003-11-26 EP disclosed
WO-2002070541-A2 PEPTIDE DEFORMYLASE INHIBITORS SMITH KLINE BEECHAM CORPORATION (US) 2002-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040087585-A1 Peptide deformylase inhibitors PDF, DPEP1, PEPD SYK 4093/4885MAPT 3406/4885CTSL 61/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.