SCHEMBL6025006

SCHEMBL6025006

COc1cc(F)c(S(=O)(=O)N2CCOCC2)cc1OC

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.63
TSHR P16473 3/20 0.62
NPSR1 Q6W5P4 1/20 0.58
KMT2A Q03164 2/20 0.57
NPC1 O15118 1/20 0.56
POLB P06746 2/20 0.54
KDM4E B2RXH2 2/20 0.52
LMNA P02545 1/20 0.52
MEN1 O00255 1/20 0.49
PKM P14618 1/20 0.49
HTT P42858 1/20 0.49
CNR1 P21554 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
BRD4 O60885 1/20 0.48
BRD2 P25440 1/20 0.48
BRD3 Q15059 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11165761 0.86 ALDH1A1 (0.54) ALDH1A1TSHRNPSR1KMT2ANPC1
SCHEMBL4468528 0.85 TSHR (0.67) ALDH1A1TSHRKMT2APOLBKDM4E
SCHEMBL6206499 0.80 CNR1 (0.52) ALDH1A1TSHRNPSR1KMT2AKDM4E
SCHEMBL1150847 0.80 TSHR (0.75) ALDH1A1TSHRNPSR1KMT2ANPC1
SCHEMBL23088183 0.77 ALDH1A1 (0.80) ALDH1A1TSHRNPSR1KMT2APOLB
SCHEMBL3345913 0.76 PKM (0.61) ALDH1A1TSHRKMT2AKDM4ELMNA
SCHEMBL20387483 0.76 NPC1 (0.70) ALDH1A1TSHRNPSR1KMT2ANPC1
SCHEMBL3408351 0.76 PKM (0.54) ALDH1A1TSHRKMT2AKDM4ELMNA
SCHEMBL29483582 0.76 NPC1 (0.70) ALDH1A1TSHRNPSR1KMT2ANPC1
SCHEMBL15120570 0.75 KMT2A (0.81) ALDH1A1TSHRNPSR1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100572375-C Spiro-benzene and dioxole and as the application of CB1 antagonist HOFFMANN LA ROCHE (CH) 2009-12-23 CN disclosed
CN-1914189-A Spiro-benzodioxoles and their use as CB1 antagonists HOFFMANN LA ROCHE (CH) 2007-02-14 CN disclosed
EP-1716132-A2 SPIRO-BENZODIOXOLES AND THEIR USE AS CB1 ANTAGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2006-11-02 EP disclosed
WO-2005075450-A2 SPIRO-BENZODIOXOLES AND THEIR USE AS CB1 ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2005-08-18 WO disclosed