SCHEMBL6027951

SCHEMBL6027951

O=C(Nc1ccccc1)c1cccc(F)c1

nearest known ligand 0.88

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.88
KMT2A Q03164 5/20 0.88
NPC1 O15118 5/20 0.88
RAB9A P51151 5/20 0.88
KCNK3 O14649 4/20 0.87
HPGD P15428 1/20 0.81
L3MBTL1 Q9Y468 1/20 0.73
KCNK9 Q9NPC2 3/20 0.69
KDM4E B2RXH2 1/20 0.69
CASP3 P42574 1/20 0.69
SENP7 Q9BQF6 1/20 0.69
SENP6 Q9GZR1 1/20 0.69
MAPT P10636 2/20 0.68
HDAC1 Q13547 2/20 0.67
HDAC6 Q9UBN7 2/20 0.67
HDAC2 Q92769 1/20 0.67
HDAC8 Q9BY41 1/20 0.67
LMNA P02545 2/20 0.64
KCNQ3 O43525 1/20 0.63
KCNQ2 O43526 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30643220 1.00 MEN1 (0.88) MEN1KMT2ANPC1RAB9AKCNK3
SCHEMBL23447715 0.89 NPC1 (1.00) MEN1KMT2ANPC1RAB9AKCNK3
SCHEMBL30739642 0.89 KMT2A (0.86) MEN1KMT2ANPC1RAB9AKCNK3
SCHEMBL1811680 0.88 L3MBTL1 (0.82) MEN1KMT2ANPC1RAB9AKCNK3
SCHEMBL6802691 0.88 KMT2A (0.78) MEN1KMT2ANPC1RAB9AKCNK3
Hydrochloric Acid SCHEMBL2106088 0.87 L3MBTL1 (0.80) MEN1KMT2ANPC1RAB9AKCNK3
SCHEMBL8374911 0.87 HDAC1 (0.85) MEN1KMT2ANPC1RAB9AKCNK3
SCHEMBL5375629 0.86 NPC1 (0.72) MEN1KMT2ANPC1RAB9AKCNK3
SCHEMBL8770869 0.86 KMT2A (0.72) MEN1KMT2ANPC1RAB9AKCNK3
SCHEMBL5168239 0.86 PGR (0.72) MEN1KMT2ANPC1RAB9AKCNK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109180518-B Secondary/tertiary amide compound and synthesis method thereof 陕西科技大学 2021-05-18 CN disclosed
CN-109180518-A Secondary/teritary amide class the compound of one kind and its synthetic method 陕西科技大学 2019-01-11 CN disclosed
EP-2757885-A1 CERTAIN CHEMICAL ENTITES, COMPOSITIONS, AND METHODS Neupharma, Inc. (US) 2014-07-30 EP disclosed
WO-2013043935-A1 CERTAIN CHEMICAL ENTITES, COMPOSITIONS, AND METHODS NEUPHARMA, INC. (US) 2013-03-28 WO disclosed
EP-1677786-A1 5-SUBSTITUTED 2-(PHENYLMETHYL)THIO-4-PHENYL-4H-1,2,4-TRIAZOLE DERIVATIVES AND RELATED COMPOUNDS AS GABA-AGONISTS FOR THE TREATMENT OF URINARY INCONTINENCE AND RELATED DISEASES Bayer HealthCare AG (DE) 2006-07-12 EP disclosed
WO-2005039569-A1 5-SUBSTITUTED 2-(PHENYLMETHYL) THIO-4-PHENYL-4H-1,2,4-TRIAZOLE DERIVATIVES AND RELATED COMPOUNDS AS GABA-AGONISTS FOR THE TREATMENT OF URINARY INCONTINENCE AND RELATED DISEASES BAYER HEALTHCARE AG (DE) 2005-05-06 WO disclosed