SCHEMBL6029004

SCHEMBL6029004

COc1cc(-c2cnc(OCC(=O)NC(Cc3ccc(Cl)c(Cl)c3)C3CCCNC3)nc2)cc(OC)c1OC

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.39
OPRK1 P41145 1/20 0.39
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
CCR3 P51677 1/20 0.37
AKT1 P31749 2/20 0.36
CDK2 P24941 1/20 0.36
IKBKB O14920 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
FYN P06241 1/20 0.34
CXCR6 O00574 1/20 0.34
MELK Q14680 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
CDK9 P50750 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6029200 0.92 ROCK2 (0.38) ROCK2ROCK1AKT1CDK2IKBKB
SCHEMBL6029151 0.89 CHEK1 (0.39) MAPK1ROCK2ROCK1AKT1CDK2
SCHEMBL6029125 0.89 MAPK1 (0.38) MAPK1OPRK1ROCK2ROCK1CCR3
SCHEMBL7827088 0.88 DYRK1A (0.39) ROCK2ROCK1AKT1CDK2IKBKB
SCHEMBL6030392 0.87 CHEK1 (0.41) AKT1CDK2CDK9
SCHEMBL6029349 0.87 MAPK1 (0.38) MAPK1OPRK1ROCK2ROCK1TP53
SCHEMBL7829880 0.84 AKT1 (0.42) ROCK2ROCK1AKT1IKBKBSLC6A2
Hydrochloric Acid SCHEMBL7833338 0.84 AKT1 (0.42) ROCK2ROCK1AKT1IKBKBSLC6A2
SCHEMBL6028227 0.82 LMNA (0.41) MAPK1ROCK2ROCK1TP53MAPT
SCHEMBL6029616 0.81 CDK2 (0.37) ROCK2ROCK1AKT1CDK2CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6984643-B2 2,5-substituted pyrimidine derivatives-CCR-3 receptor antagonists ROCHE PALO ALTO LLC (US) 2006-01-10 US disclosed