SCHEMBL6029349

SCHEMBL6029349

COc1cc(-c2cnc(OCC(=O)NC(Cc3cccc(Cl)c3Cl)C3CCCNC3)nc2)cc(OC)c1OC

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.38
OPRK1 P41145 1/20 0.38
CDK9 P50750 5/20 0.37
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
SLC6A2 P23975 5/20 0.35
SLC6A4 P31645 5/20 0.35
SLC6A3 Q01959 4/20 0.35
CYP2D6 P10635 2/20 0.35
KCNH2 Q12809 2/20 0.35
CXCR6 O00574 3/20 0.35
TP53 P04637 1/20 0.34
MELK Q14680 2/20 0.34
RXFP1 Q9HBX9 1/20 0.34
CYP3A4 P08684 1/20 0.34
CCNT1 O60563 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6029742 0.93 CDK9 (0.38) CDK9ROCK2ROCK1SLC6A2SLC6A4
SCHEMBL6029579 0.89 MAPK1 (0.37) MAPK1OPRK1CDK9ROCK2ROCK1
SCHEMBL6028513 0.89 GRIN1 (0.41) CDK9SLC6A2SLC6A4TP53CYP3A4
SCHEMBL6030272 0.89 CHEK1 (0.37) MAPK1CDK9SLC6A2SLC6A4SLC6A3
SCHEMBL6029004 0.87 MAPK1 (0.39) MAPK1OPRK1CDK9ROCK2ROCK1
SCHEMBL7826595 0.84 SLC6A4 (0.39) ROCK2ROCK1SLC6A2SLC6A4SLC6A3
SCHEMBL6030139 0.82 ALOX15 (0.37) CDK9ROCK2SLC6A2SLC6A4SLC6A3
SCHEMBL7831249 0.80 SLC6A4 (0.38) OPRK1SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL6029200 0.79 ROCK2 (0.38) CDK9ROCK2ROCK1RXFP1CCNT1
SCHEMBL6028530 0.79 CHEK1 (0.37) CDK9SLC6A2SLC6A4SLC6A3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6984643-B2 2,5-substituted pyrimidine derivatives-CCR-3 receptor antagonists ROCHE PALO ALTO LLC (US) 2006-01-10 US disclosed