SCHEMBL6032802

SCHEMBL6032802

CCOC(=O)c1cccnc1I

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.59
HTT P42858 1/20 0.55
ALDH1A1 P00352 4/20 0.51
HSD17B10 Q99714 2/20 0.51
L3MBTL1 Q9Y468 3/20 0.50
TP53 P04637 1/20 0.49
BRD4 O60885 1/20 0.49
POLB P06746 2/20 0.47
TBXAS1 P24557 1/20 0.47
MAPK1 P28482 1/20 0.47
PDE4A P27815 1/20 0.47
ELANE P08246 2/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CYP1A2 P05177 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL109206 0.83 TSHR (0.63) TSHRHTTALDH1A1HSD17B10L3MBTL1
SCHEMBL29571304 0.83 TSHR (0.63) TSHRHTTALDH1A1HSD17B10L3MBTL1
SCHEMBL29870373 0.81 BRD4 (0.61) TSHRHTTALDH1A1HSD17B10L3MBTL1
SCHEMBL162019 0.81 TSHR (0.61) TSHRHTTALDH1A1HSD17B10L3MBTL1
SCHEMBL1737254 0.81 BRD4 (0.61) TSHRHTTALDH1A1HSD17B10L3MBTL1
SCHEMBL6043587 0.81 TSHR (0.61) TSHRHTTALDH1A1HSD17B10L3MBTL1
SCHEMBL1807370 0.81 TDP1 (0.55) TSHRHTTALDH1A1HSD17B10L3MBTL1
SCHEMBL12897074 0.80 TSHR (0.59) TSHRHTTALDH1A1HSD17B10L3MBTL1
SCHEMBL49913 0.80 POLB (0.66) TSHRHTTALDH1A1L3MBTL1POLB
Hydrochloric Acid SCHEMBL4990673 0.80 TSHR (0.59) TSHRHTTALDH1A1HSD17B10L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104945316-B A kind of method of microwave method synthesis 2- halos nicotinate and its intermediate 山东师范大学 2018-05-04 CN claimed
CN-104945317-B A kind of method of supercritical ultrasonics technology synthesis 2- halos nicotinate and its intermediate 山东师范大学 2018-03-30 CN claimed
CN-107540605-A For hair or the choline ester type compound of scalp care 李明霞 2018-01-05 CN claimed
CN-106349157-B A kind of method of hydro-thermal method synthesis 2- halogenated nicotinate and the halogenated niacin of 2- 山东华阳农药化工集团有限公司 2019-02-01 CN disclosed
CN-107540605-A For hair or the choline ester type compound of scalp care 李明霞 2018-01-05 CN disclosed
CN-106349157-A Method using hydrothermal method to synthesize 2-halogeneated nicotinate and 2-halogeneated nicotinic acid 山东华阳农药化工集团有限公司 2017-01-25 CN disclosed
US-6992094-B1 Diarylselenide compounds and their use in human or veterinary medicine and in cosmetics GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2006-01-31 US disclosed
US-20060014803-A1 Diarylselenide compounds and their use in human or veterinary medicine and in cosmetics GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2006-01-19 US disclosed
US-5672710-A SPECIFIC AGONISTS FOR THE RXR RETINOID RECEPTOR RATHER THAN THE RAR ONE; SIDE EFFECT REDUCTION; SKIN AND NERVOUS SYTEM DISORDERS; ANTICARCINOGENIC AGENTS; VISION DEFECTS ALLERGAN (US) 1997-09-30 US disclosed
US-5670456-A Compounds SANDOZ LTD. (CH) 1997-09-23 US disclosed
WO-1997016422-A1 SULFIDES, SULFOXIDES AND SULFONES DISUBSTITUTED WITH A TETRAHYDRONAPHTHALENYL, CHROMANYL, THIOCHROMANYL OR TETRAHYDROQUINOLINYL AND SUBSTITUTED PHENYL OR HETEROARYL GROUP, HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN (US) 1997-05-09 WO disclosed
US-5506191-A Heterocyclic hydrazines and hydrazones SANDOZ LTD. (CH) 1996-04-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060014803-A1 Diarylselenide compounds and their use in human or veterinary medicine and in cosmetics TYR, DERL1, GPX1 TSHR 2188/4885HTT 536/4885ALDH1A1 118/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.