SCHEMBL49913

SCHEMBL49913

CCOC(=O)c1cccnc1Cl

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.66
L3MBTL1 Q9Y468 2/20 0.64
LMNA P02545 3/20 0.63
CYP2C19 P33261 3/20 0.62
CYP1A2 P05177 2/20 0.62
CYP2C9 P11712 2/20 0.62
CASP3 P42574 1/20 0.62
SENP8 Q96LD8 1/20 0.62
SENP7 Q9BQF6 1/20 0.62
SENP6 Q9GZR1 1/20 0.62
KMT2A Q03164 5/20 0.59
MEN1 O00255 4/20 0.59
TSHR P16473 1/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
ALDH1A1 P00352 1/20 0.59
TDP1 Q9NUW8 3/20 0.58
CYP2D6 P10635 1/20 0.58
PKM P14618 1/20 0.58
HTT P42858 2/20 0.57
AGTR1 P30556 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3584951 0.98 POLB (0.64) POLBL3MBTL1LMNACYP2C19CYP1A2
SCHEMBL28348218 0.90 TSHR (0.60) POLBL3MBTL1LMNACYP2C19CYP1A2
SCHEMBL5532922 0.86 POLB (0.51) POLBL3MBTL1LMNACYP2C19CYP1A2
Niacin SCHEMBL6418540 0.85 CYP2C9 (0.58) POLBL3MBTL1LMNACYP2C19CYP1A2
SCHEMBL30609724 0.84 L3MBTL1 (0.64) POLBL3MBTL1LMNACYP2C19CYP1A2
SCHEMBL28350930 0.84 TP53 (0.63) POLBL3MBTL1LMNAKMT2AMEN1
SCHEMBL28351060 0.83 POLB (0.58) POLBL3MBTL1LMNACYP2C19CYP1A2
SCHEMBL109206 0.83 TSHR (0.63) L3MBTL1CYP1A2TSHRSMN1; SMN2ALDH1A1
SCHEMBL29571304 0.83 TSHR (0.63) L3MBTL1CYP1A2TSHRSMN1; SMN2ALDH1A1
SCHEMBL7954798 0.83 ALDH1A1 (0.63) POLBL3MBTL1LMNACYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 779 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10035768-B2 C5aR antagonists CHEMOCENTRYX, INC. (US) 2018-07-31 US claimed
US-20180179160-A1 C5AR ANTAGONISTS CHEMOCENTRYX, INC. 2018-06-28 US claimed
EP-3078658-A1 C5AR ANTAGONISTS ChemoCentryx, Inc. (US) 2016-10-12 EP claimed
US-5248781-A Preparation of substituted anilino-nicotinic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1993-09-28 US claimed
US-12637467-B2 Inhibitor of BTK and mutants thereof NEWAVE PHARMACEUTICAL INC. (US) 2026-05-26 US disclosed
US-20260132127-A1 NOVEL SPIRO COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2026-05-14 US disclosed
US-20260125364-A1 HETEROAROMATIC COMPOUNDS AND THEIR USE AS DOPAMINE D1 LIGANDS PFIZER (US) 2026-05-07 US disclosed
CN-121779321-A Industrial production method of 2-chloronicotinic acid 江苏三鹏生物化工有限公司 2026-04-03 CN disclosed
CN-120790068-A Continuous production device and production method for 2-chloronicotinic acid 苏利(宁夏)新材料科技有限公司 2025-10-17 CN disclosed
US-20250236897-A1 PROCESSES FOR PREPARATION OF AVACOPAN AND INTERMEDIATES THEREOF TEVA PHARMACEUTICALS INTERNATIONAL GMBH (CH) 2025-07-24 US disclosed
US-20250213547-A1 METHODS OF TREATING NEUROLOGICAL DISEASES TAKEDA PHARMACEUTICALS CO (JP) 2025-07-03 US disclosed
CN-115710217-B Flunixin meglumine synthesis method suitable for industrial production 江苏恒盛药业有限公司 2025-06-13 CN disclosed
US-4740511-A ANTIALLERGENS, ANTIINFLAMMATORY, ANTIULCER AGENTS SCHERING CORPORATION (US) 1988-04-26 US disclosed
US-4680298-A Tricyclic anti-allergy and use as anti-inflammatory agents SCHERING CORPORATION (US) 1987-07-14 US disclosed
US-4632923-A Substituted hetero spiro pyridine derivatives as anti-allergy and anti-inflammatory agents SCHERING CORPORATION (US) 1986-12-30 US disclosed
CN-85106252-A The preparation method of compound and application thereof 1986-06-10 CN disclosed
EP-0174717-A1 Benzimidazoles, and their production formulation and use as gastric acid secretion inhibitors FISONS plc (GB) 1986-03-19 EP disclosed
EP-0144996-A2 Substituted spiro pyridine derivatives, pharmaceutical compositions containing them and processes for the preparation of such compounds and compositions SCHERING CORPORATION (US) 1985-06-19 EP disclosed
EP-0127135-A2 Fused tricyclic derivatives of naphthyridinone and pyridone and the corresponding thiones SCHERING CORPORATION (US) 1984-12-05 EP disclosed
US-4205073-A Anti-diarrheal anilino nicotinic acids and method of using same SCHERING CORPORATION (US) 1980-05-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250236897-A1 PROCESSES FOR PREPARATION OF AVACOPAN AND INTERMEDIATES THEREOF DHPS, VARS1, AGPS POLB 158/4885L3MBTL1 4637/4885LMNA 1946/4885
US-20260125364-A1 HETEROAROMATIC COMPOUNDS AND THEIR USE AS DOPAMINE D1 LIGANDS HTR6, HTR3C, OPRD1 POLB 1831/4885L3MBTL1 783/4885LMNA 2257/4885
US-20180179160-A1 C5AR ANTAGONISTS C5AR1, C5AR2, C3AR1 POLB 3658/4885L3MBTL1 2243/4885LMNA 2969/4885
US-10035768-B2 C5aR antagonists C5AR1, C5AR2, C3AR1 POLB 3658/4885L3MBTL1 2243/4885LMNA 2969/4885
US-20250213547-A1 METHODS OF TREATING NEUROLOGICAL DISEASES SMN1; SMN2, PMP22, GBA2 POLB 2602/4885L3MBTL1 2698/4885LMNA 2937/4885
US-12637467-B2 Inhibitor of BTK and mutants thereof BTK, CNKSR1, SYK POLB 1177/4885L3MBTL1 384/4885LMNA 3447/4885
US-20260132127-A1 NOVEL SPIRO COMPOUND TRHR, NR3C2, THRB POLB 4761/4885L3MBTL1 3822/4885LMNA 2025/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.