SCHEMBL6038763

SCHEMBL6038763

CNC(=O)n1ccc2ccc(Oc3ccnc(OC(=O)NC(=O)Oc4ccccc4)c3)cc21

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GCK P35557 1/20 0.40
RAF1 P04049 1/20 0.37
BRAF P15056 1/20 0.37
FGFR1 P11362 15/20 0.37
PPARG P37231 2/20 0.37
FGF2 P09038 1/20 0.36
FGFR4 P22455 1/20 0.36
FGFR3 P22607 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6038705 0.89 KDR (0.41) PPARG
SCHEMBL6517430 0.85 GCK (0.37) GCKRAF1BRAFFGFR1PPARG
SCHEMBL5101452 0.81 GCK (0.40) GCKRAF1BRAFFGFR1FGF2
SCHEMBL6038760 0.80 GCK (0.39) GCKRAF1BRAFFGFR1FGF2
SCHEMBL6038815 0.79 ASAH1 (0.37) FGFR1PPARG
SCHEMBL5107824 0.78 GCK (0.53) GCKFGFR1FGF2FGFR4FGFR3
SCHEMBL6038529 0.78 RAB9A (0.39)
SCHEMBL6038451 0.78 MCHR1 (0.38)
SCHEMBL6038635 0.78 KDR (0.36)
SCHEMBL5101352 0.78 FGFR1 (0.42) FGFR1FGF2FGFR4FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060004029-A1 Nitrogen-containing aromatic derivatives EISAI R&D MANAGEMENT CO., LTD. (JP) 2006-01-05 US disclosed
EP-1522540-A1 AZAARENE DERIVATIVES Eisai Co., Ltd. (JP) 2005-04-13 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060004029-A1 Nitrogen-containing aromatic derivatives NR0B2, NR0B1, NR4A1 GCK 3607/4885RAF1 1150/4885BRAF 1488/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.