1-Methylimidazole

1-Methylimidazole

SCHEMBL6040916

CNC(=O)c1ccc[nH]1.Cn1ccnc1

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD38 P28907 1/20 0.42
NFKB1 P19838 1/20 0.42
QPCT Q16769 1/20 0.42
HSD17B10 Q99714 1/20 0.42
QPCTL Q9NXS2 1/20 0.42
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
TBXAS1 P24557 1/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
GFER P55789 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ATM Q13315 1/20 0.38
TMIGD3 P0DMS9 1/20 0.37
ADORA1 P30542 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14742539 0.82 KDM4E (0.44) KDM4ENPC1RAB9AGFERATM
SCHEMBL888653 0.80
SCHEMBL28029054 0.78
SCHEMBL8376540 0.71 DRD2 (0.42) NPC1RAB9AGFERALDH1A1LMNA
1-Methylimidazole SCHEMBL28947361 0.67 NFKB1 (0.75) NFKB1QPCTHSD17B10QPCTLTBXAS1
1-Methylimidazole SCHEMBL19356956 0.67 NFKB1 (0.75) NFKB1QPCTHSD17B10QPCTLTBXAS1
1-Methylimidazole SCHEMBL27892740 0.67 NFKB1 (0.94) NFKB1QPCTHSD17B10QPCTLTBXAS1
1-Methylimidazole SCHEMBL8719680 0.67
Benzoic Acid SCHEMBL2804715 0.66 NFKB1 (0.54) NFKB1QPCTHSD17B10QPCTLTBXAS1
Phthalic Acid SCHEMBL12076342 0.66 NFKB1 (0.54) NFKB1QPCTHSD17B10QPCTLTBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170313747-A1 SELF-ASSEMBLED NANOSTRUCTURES DOE-DEITR 2017-11-02 US disclosed
US-9650421-B2 Self-assembled nanostructures NORTHWESTERN UNIVERSITY (US) 2017-05-16 US disclosed
US-20150031127-A1 SELF-ASSEMBLED NANOSTRUCTURES NORTHWESTERN UNIVERSITY (US) 2015-01-29 US disclosed
EP-1599474-B1 Heterocyclic oligomeric compounds for DNA recognition CALIFORNIA INST OF TECHN (US) 2013-04-24 EP disclosed
WO-2013033658-A1 SELF-ASSEMBLED NANOSTRUCTURES NORTHWESTERN UNIVERSITY (US) 2013-03-07 WO disclosed
US-7087378-B1 Design, synthesis and use of specific polyamide DNA-binding ligands CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2006-08-08 US disclosed
US-6472537-B1 POLYMERS FROM PRIMARY AMINE AND CARBOXYLIC ACID SUBSTITUTED PYROLE, HYDROXYPYROLE AND IMIDAZOLE MONOMERS AND HAVING 4-AMINOBUTYRIC ACID LINKER FORMING HAIRPIN TURNS AND OPTION-ALLY AMINO ACID RESIDUES; BINDING TO SPECIFIC CALIFORNIA INSTITUTE OF TECHNOLOGY 2002-10-29 US disclosed
EP-0973740-A1 DESIGN, SYNTHESIS AND USE OF SPECIFIC POLYAMIDE DNA-BINDING LIGANDS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2000-01-26 EP disclosed
EP-0968186-A1 IMPROVED POLYAMIDES FOR BINDING IN THE MINOR GROOVE OF DOUBLE STRANDED DNA CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2000-01-05 EP disclosed
WO-1998037066-A9 IMPROVED POLYAMIDES FOR BINDING IN THE MINOR GROOVE OF DOUBLE STRANDED DNA 1999-02-04 WO disclosed
WO-1998037067-A1 DESIGN, SYNTHESIS AND USE OF SPECIFIC POLYAMIDE DNA-BINDING LIGANDS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 1998-08-27 WO disclosed
WO-1998037066-A1 IMPROVED POLYAMIDES FOR BINDING IN THE MINOR GROOVE OF DOUBLE STRANDED DNA CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 1998-08-27 WO disclosed