SCHEMBL6045133

SCHEMBL6045133

[CH2]c1ccc(C#Cc2ccc(Cl)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.47
KCNH2 Q12809 3/20 0.47
LMNA P02545 2/20 0.42
CYP2A6 P11509 1/20 0.42
APP P05067 2/20 0.38
MAOA P21397 2/20 0.37
MAOB P27338 2/20 0.37
ACACB O00763 1/20 0.36
ADK P55263 2/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
IDO1 P14902 1/20 0.33
HAO1 Q9UJM8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20015814 0.86 LMNA (0.57) GRM5KCNH2LMNACYP2A6APP
SCHEMBL719360 0.86 LMNA (0.57) GRM5KCNH2LMNACYP2A6APP
Charcoal, Activated SCHEMBL31286310 0.83 KCNH2 (0.54) GRM5KCNH2LMNACYP2A6APP
SCHEMBL40632 0.83
SCHEMBL6606391 0.80
SCHEMBL29142535 0.80
Hydrochloric Acid SCHEMBL28508743 0.80
SCHEMBL4946113 0.76 APP (0.67) GRM5KCNH2LMNAAPP
SCHEMBL717633 0.76 APP (0.67) GRM5KCNH2LMNACYP2A6APP
SCHEMBL4452235 0.76 LMNA (0.44) GRM5KCNH2LMNACYP2A6APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7109377-B2 Synthesis of combinatorial libraries of compounds reminiscent of natural products PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2006-09-19 US disclosed
US-6448443-B1 GENERATED FROM DIVERSIFIABLE SCAFFOLDS SYNTHESIZED FROM THE PYRIDINE-BASED TEMPLATE ISONICOTINAMIDE; ALSO PROVIDES A NOVEL ORTHO-NITROBENZYL PHOTOLINKER; SYNTHESIZED FROM A SHIKIMIC ACID BASED EPOXYOL TEMPLATE PRESIDENT AND FELLOWS OF HARVARD COLLEGE 2002-09-10 US disclosed