SCHEMBL6047660

SCHEMBL6047660

COC1=CC[CH]C(c2cccc(OC)c2)=C1c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
DYRK1A Q13627 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
ALOX5 P09917 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2B6 P20813 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887285 0.91 ALKBH3 (0.44) ALDH1A1MAPTNPSR1NPC1TP53
SCHEMBL6047606 0.84 NR1I3 (0.39) MAPTNPC1TP53NFKB1RAB9A
SCHEMBL5887303 0.84 CASR (0.39) MAPTSMN1; SMN2ALOX5HTR1AGSK3B
SCHEMBL5887353 0.79 MEN1 (0.35) NPC1TP53RAB9ASMN1; SMN2CLK4
SCHEMBL5887155 0.78 NOTUM (0.36) MAPTNPC1SMN1; SMN2ALOX5NR1I3
SCHEMBL5887199 0.76 KMT2A (0.35) ALDH1A1NPC1TP53RAB9ASMN1; SMN2
SCHEMBL5887105 0.76 ESR2 (0.35) MAPTNPC1TP53SMN1; SMN2ALOX5
SCHEMBL5887499 0.73 ALKBH3 (0.41) ALDH1A1MAPTNPSR1NPC1TP53
SCHEMBL5887320 0.72 ACHE (0.33) NPC1RAB9AALOX5CYP2C9CYP2D6
SCHEMBL5887750 0.72 MAPK10 (0.38) MAPTNR1I3HTR1ACYP2A6GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed