SCHEMBL6048146

SCHEMBL6048146

CC[C@@H](NC(=O)[CH]C[Si](C)(C)C)C(=O)c1nc2ccccc2o1

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSS P25774 19/20 0.50
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5519481 0.90 CTSS (0.48) CTSSCYP3A4CYP2C9
SCHEMBL5517725 0.90 CTSS (0.48) CTSSCYP3A4CYP2C9
SCHEMBL27663441 0.83 CTSS (0.57) CTSSCYP3A4CYP2C9
SCHEMBL3877756 0.82 CTSS (0.47) CTSSCYP3A4CYP2C9
SCHEMBL5519871 0.82 FAAH (0.43) CTSSCYP3A4CYP2C9
SCHEMBL5520458 0.82 FAAH (0.43) CTSSCYP3A4CYP2C9
SCHEMBL6048147 0.81 CTSS (0.51) CTSSCYP3A4CYP2C9
SCHEMBL5517452 0.80 FAAH (0.46) CTSSCYP3A4CYP2C9
SCHEMBL14378277 0.80 CTSS (0.51) CTSSCYP3A4CYP2C9
SCHEMBL14378197 0.80 CTSS (0.51) CTSSCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716158-A2 SILINANE COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS Schering Aktiengesellschaft (DE) 2006-11-02 EP disclosed
WO-2005074904-A2 SILINANE COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 2005-08-18 WO disclosed