SCHEMBL60518

SCHEMBL60518

CC(=O)O[C@]1(C(C)=O)[C@H](O)[C@@H](CO)O[C@@]1(C(C)=O)n1ccc(=O)[nH]c1=O

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC28A1 O00337 1/20 0.39
SLC28A2 O43868 1/20 0.39
SLC29A1 Q99808 1/20 0.39
SLC28A3 Q9HAS3 1/20 0.39
P2RY6 Q15077 8/20 0.33
P2RY14 Q15391 3/20 0.33
P2RY2 P41231 3/20 0.31
P2RY4 P51582 2/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
OGT O15294 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2337871 0.84 SLC28A1 (0.41) SLC28A1SLC28A2SLC29A1SLC28A3P2RY6
SCHEMBL2337859 0.84 SLC28A1 (0.41) SLC28A1SLC28A2SLC29A1SLC28A3P2RY6
SCHEMBL6136114 0.82 SLC28A1 (0.42) SLC28A1SLC28A2SLC29A1SLC28A3P2RY6
SCHEMBL28148332 0.82 TK1 (0.37) ALDH1A1LMNA
SCHEMBL29134987 0.81 TK2 (0.35)
SCHEMBL9237885 0.80 LMNA (0.37) LMNA
SCHEMBL381848 0.79 PDE3A (0.41) SLC29A1ALDH1A1LMNA
SCHEMBL28289547 0.77 TK2 (0.46)
SCHEMBL12813023 0.75 DNMT1 (0.41) ALDH1A1LMNA
SCHEMBL1285619 0.75 POLB (0.39) SLC28A1SLC28A2SLC29A1SLC28A3P2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 9418 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
US-20240343697-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2024-10-17 US claimed
WO-2024162590-A1 COMPOSITION FOR PREVENTING OR TREATING PROSTATIC HYPERTROPHY, CONTAINING, AS ACTIVE INGREDIENTS, SALVIA MILTIORRHIZA BUNGE EXTRACT, METAL MINERAL DIAMINATE AND URIDINE 주식회사 건강중심주의 2024-08-08 WO claimed
US-11345956-B2 Methods and compositions related to prostate cancer therapeutics THE JOHNS HOPKINS UNIVERSITY (US) 2022-05-31 US claimed
CN-112301118-B Method and kit for simultaneously obtaining RNA abundance and active RNA polymerase sites in full transcriptome range 浙江大学 2022-05-13 CN claimed
WO-2021261855-A1 ZINC TRANSPORTER ACTIVATOR COMPOSITION 주식회사 메타센테라퓨틱스 2021-12-30 WO claimed
US-11207289-B2 Use of benzofuran lignans to induce IL-25 expression and suppress mammary tumor metastasis ACADEMIA SINICA (TW) 2021-12-28 US claimed
US-20210154200-A1 7-BENZYL-4-(METHYLBENZYL)-2,4,6,7,8,9-HEXAHYDROIMIDAZO[1,2-A]PYRIDO[3,4-E]PYRIMIDIN-5 (1H)-ONE, SALTS THEREOF AND METHODS OF USING THE SAME IN COMBINATION THERAPY ONCOCEUTICS, INC. (US) 2021-05-27 US claimed
US-10953073-B2 XTEN conjugate compositions and methods of making same AMUNIX PHARMACEUTICALS, INC. (US) 2021-03-23 US claimed
WO-1996040165-A1 METHODS OF REDUCING TOXICITY OF CHEMOTHERAPEUTIC AND ANTIVIRAL AGENTS WITH ACYLATED PYRIMIDINE NUCLEOSIDES PRO-NEURON, INC. (US) 1996-12-19 WO claimed
WO-1996001115-A1 PYRIMIDINE NUCLEOTIDE PRECURSORS FOR TREATMENT OF SYSTEMIC INFLAMMATION AND INFLAMMATORY HEPATITIS PRO-NEURON, INC. (US) 1996-01-18 WO claimed
EP-0594667-A4 TREATMENT OF CHEMOTHERAPEUTIC AGENT AND ANTIVIRAL AGENT TOXICITY WITH ACYLATED PYRIMIDINE NUCLEOSIDES PRO NEURON INC (US) 1996-01-10 EP claimed
EP-0679160-A1 PYRIMIDINE NUCLEOTIDE PRECURSORS FOR TREATMENT OF SYSTEMIC INFLAMMATION AND INFLAMMATORY HEPATITIS PRO-NEURON, INC. (US) 1995-11-02 EP claimed
WO-1994026761-A1 TREATMENT OF CHEMOTHERAPEUTIC AGENT AND ANTIVIRAL AGENT TOXICITY WITH ACYLATED PYRIMIDINE NUCLEOSIDES PRO-NEURON, INC. (US) 1994-11-24 WO claimed
CN-1095268-A Pyrimidine nucleotide precursors for the treatment of systemic inflammation and inflammatory hepatitis PRO NEURON INC (US) 1994-11-23 CN claimed
WO-1994013687-A1 PYRIMIDINE NUCLEOTIDE PRECURSORS FOR TREATMENT OF SYSTEMIC INFLAMMATION AND INFLAMMATORY HEPATITIS PRO-NEURON, INC. (US) 1994-06-23 WO claimed
EP-0594667-A1 TREATMENT OF CHEMOTHERAPEUTIC AGENT AND ANTIVIRAL AGENT TOXICITY WITH ACYLATED PYRIMIDINE NUCLEOSIDES PRO-NEURON, INC. (US) 1994-05-04 EP claimed
CN-1071577-A Handle the toxicity of chemotherapy reagent and Anti-virus agent with acylated pyrimidine nucleosides PRO NEURON INC (US) 1993-05-05 CN claimed
WO-1993001202-A1 TREATMENT OF CHEMOTHERAPEUTIC AGENT AND ANTIVIRAL AGENT TOXICITY WITH ACYLATED PYRIMIDINE NUCLEOSIDES PRO-NEURON, INC. (US) 1993-01-21 WO claimed