SCHEMBL6059152

SCHEMBL6059152

CC(C)(C)OC(=O)Nc1ncc(CO)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STK17B O94768 1/20 0.42
STK17A Q9UEE5 1/20 0.42
MAPKAPK2 P49137 3/20 0.41
ALDH1A1 P00352 2/20 0.40
LCK P06239 1/20 0.40
ATR Q13535 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 1/20 0.38
CYP17A1 P05093 1/20 0.37
NAMPT P43490 1/20 0.37
POLB P06746 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
NR4A1 P22736 1/20 0.36
MAPT P10636 1/20 0.36
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6058971 0.88 STK17B (0.41) STK17BSTK17AMAPKAPK2ALDH1A1ATR
SCHEMBL13428494 0.84 STK17B (0.54) STK17BSTK17AALDH1A1L3MBTL1TDP1
SCHEMBL6059338 0.83 LCK (0.40) STK17BSTK17AMAPKAPK2LCKATR
SCHEMBL6059446 0.81 CPB2 (0.41) STK17BSTK17AMAPKAPK2ALDH1A1L3MBTL1
SCHEMBL9646590 0.80 ALDH1A1 (0.46) ALDH1A1L3MBTL1TDP1MEN1KMT2A
SCHEMBL14822488 0.80 ATR (0.40) STK17BSTK17AMAPKAPK2ALDH1A1ATR
SCHEMBL6060000 0.79 CPB2 (0.39) STK17BSTK17AMAPKAPK2ALDH1A1L3MBTL1
SCHEMBL6059420 0.79 L3MBTL1 (0.38) STK17BSTK17AMAPKAPK2ALDH1A1ATR
SCHEMBL7382657 0.78 NR4A1 (0.39) STK17BSTK17AMAPKAPK2ALDH1A1ATR
Malonic Acid Diethyl Ester SCHEMBL7380709 0.78 L3MBTL1 (0.41) STK17BSTK17AMAPKAPK2ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7071175-B1 Pyridine mercapto carboxylic acids as carboxypeptidase U inhibitors ASTRAZENECA AB (SE) 2006-07-04 US disclosed
EP-1180098-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2002-02-20 EP disclosed
WO-2000066557-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2000-11-09 WO disclosed