SCHEMBL6061967

SCHEMBL6061967

CS(=O)(=O)N=CN[C@@H](CC1CCCCC1)C(=O)NCCC[C@H](O)c1nc2ccccc2o1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSS P25774 11/20 0.46
CTSL P07711 8/20 0.40
MMP2 P08253 6/20 0.37
MMP1 P03956 5/20 0.37
MMP3 P08254 5/20 0.37
CTSK P43235 2/20 0.36
CHRNB2 P17787 2/20 0.36
CHRNB4 P30926 2/20 0.36
CHRNA3 P32297 2/20 0.36
CHRNA4 P43681 2/20 0.36
CPB2 Q96IY4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5703798 0.87 CTSS (0.44) CTSSCTSLMMP2MMP1MMP3
SCHEMBL7259493 0.85 CTSS (0.45) CTSSCTSLMMP2MMP1MMP3
SCHEMBL5946322 0.83 CTSS (0.40) CTSSCTSLCTSK
SCHEMBL5946098 0.83 CTSS (0.40) CTSSCTSLCTSK
SCHEMBL5946093 0.83 CTSS (0.40) CTSSCTSLCTSK
Hydrochloric Acid SCHEMBL7255797 0.79 CTSS (0.47) CTSSCTSLMMP2MMP1MMP3
SCHEMBL7255828 0.77 CTSS (0.48) CTSSCTSLMMP2MMP1MMP3
SCHEMBL6206920 0.74 CTSS (0.41) CTSS
SCHEMBL7260348 0.74 CTSS (0.35) CTSS
SCHEMBL7259168 0.74 CTSS (0.43) CTSSCTSLCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694357-A1 USE OF CATHEPSIN S INHIBITORS FOR TREATING AN IMMUNE RESPONSE CAUSED BY ADMINISTRATION OF A SMALL MOLECULE THERAPEUTIC OR BIOLOGIC AXYS PHARMACEUTICALS, INC. (US) 2006-08-30 EP disclosed
WO-2005058348-A1 USE OF CATHEPSIN S INHIBITORS FOR TREATING AN IMMUNE RESPONSE CAUSED BY ADMINISTRATION OF A SMALL MOLECULE THERAPEUTIC OR BIOLOGIC AXYS PHARMACEUTICALS, INC. (US) 2005-06-30 WO disclosed