SCHEMBL6065834

SCHEMBL6065834

Cn1ncc(NC([N])=O)c1NC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 2/20 0.36
NTRK1 P04629 2/20 0.35
BRD4 O60885 3/20 0.35
BRD9 Q9H8M2 3/20 0.35
KAT2B Q92831 2/20 0.35
BPTF Q12830 1/20 0.35
VNN1 O95497 1/20 0.34
KDM4C Q9H3R0 1/20 0.33
ITK Q08881 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HTT P42858 1/20 0.33
FLT1 P17948 2/20 0.32
KDR P35968 1/20 0.32
MAPK1 P28482 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3119092 0.89 LPAR1 (0.38) LPAR1NTRK1BRD4BRD9KAT2B
SCHEMBL6425412 0.88 ALDH1A1 (0.37) LPAR1NTRK1BRD4BRD9KAT2B
SCHEMBL6065837 0.88 LPAR1 (0.37) LPAR1NTRK1BRD4BRD9KAT2B
SCHEMBL3111828 0.85 NTRK1 (0.36) LPAR1NTRK1BRD4BRD9KAT2B
SCHEMBL5500962 0.85 ADRA2C (0.39) LPAR1NTRK1BRD4BRD9KAT2B
SCHEMBL6425423 0.85 HPGD (0.40) NTRK1MEN1KMT2AHTTMAPK1
SCHEMBL5497720 0.83 KDM4E (0.36) LPAR1NTRK1BRD4BRD9KAT2B
SCHEMBL3105963 0.83 ALDH1A1 (0.41) LPAR1MEN1KMT2AHTTCYP1A2
SCHEMBL4199230 0.81 BRD9 (0.36) LPAR1BRD4BRD9KAT2BBPTF
SCHEMBL6385917 0.81 NTRK1 (0.36) LPAR1NTRK1BRD4BRD9KAT2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663245-A1 CEPHEM COMPOUNDS Astellas Pharma Inc. (JP) 2006-06-07 EP disclosed
WO-2005027909-A1 CEPHEM COMPOUNDS ASTELLAS PHARMA INC. (JP) 2005-03-31 WO disclosed