SCHEMBL4199230

SCHEMBL4199230

Cn1ncc(NC=O)c1NC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRD9 Q9H8M2 8/20 0.36
KAT2B Q92831 8/20 0.36
BRD4 O60885 5/20 0.36
BPTF Q12830 2/20 0.36
KCNN4 O15554 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HIF1A Q16665 1/20 0.32
TSHR P16473 1/20 0.32
PABPC1 P11940 1/20 0.31
BRD1 O95696 1/20 0.31
ACHE P22303 1/20 0.31
BRPF1 P55201 1/20 0.31
KAT2A Q92830 1/20 0.31
BRD7 Q9NPI1 1/20 0.31
BAZ2B Q9UIF8 1/20 0.31
BRPF3 Q9ULD4 1/20 0.31
LPAR1 Q92633 1/20 0.30
VNN1 O95497 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Carbamic Acid SCHEMBL3119239 0.93 BRD4 (0.32) BRD9KAT2BBRD4BPTFALDH1A1
Carbamic Acid SCHEMBL3119184 0.93 BRD4 (0.32) BRD9KAT2BBRD4BPTFALDH1A1
SCHEMBL6065834 0.81 LPAR1 (0.36) BRD9KAT2BBRD4BPTFLPAR1
SCHEMBL4199889 0.81 GAA (0.32)
SCHEMBL3119092 0.81 LPAR1 (0.38) BRD9KAT2BBRD4BPTFALDH1A1
SCHEMBL4205063 0.80 ALDH1A1 (0.36) BRD9KAT2BBRD4BPTFKCNN4
SCHEMBL6065837 0.80 LPAR1 (0.37) BRD9KAT2BBRD4BPTFALDH1A1
SCHEMBL6425412 0.80 ALDH1A1 (0.37) BRD9KAT2BBRD4BPTFALDH1A1
SCHEMBL5500962 0.76 ADRA2C (0.39) BRD9KAT2BBRD4BPTFLPAR1
SCHEMBL6425423 0.76 HPGD (0.40) ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1556389-B9 CEPHEM COMPOUNDS ASTELLAS PHARMA INC (JP) 2015-09-09 EP disclosed
EP-1556389-B3 CEPHEM COMPOUNDS ASTELLAS PHARMA INC (JP) 2015-04-01 EP disclosed
US-20090012054-A1 Cephem Compounds and Use as Antimicrobial Agents ASTELLAS PHARMA INC. (JP) 2009-01-08 US disclosed
EP-1994035-A1 CEPHEM COMPOUNDS AND USE AS ANTIMICROBIAL AGENTS Astellas Pharma Inc. (JP) 2008-11-26 EP disclosed
WO-2007119511-A1 CEPHEM COMPOUNDS AND USE AS ANTIMICROBIAL AGENTS ASTELLAS PHARMA INC. (JP) 2007-10-25 WO disclosed
CN-100343260-C Cephem compounds FUJISAWA PHARMACEUTICAL CO (JP) 2007-10-17 CN disclosed
EP-1556389-B1 CEPHEM COMPOUNDS ASTELLAS PHARMA INC (JP) 2007-07-25 EP disclosed
US-20070037786-A1 Cephem compounds WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2007-02-15 US disclosed
US-7129232-B2 For therapy of of infectious diseases ASTELLAS PHARMA INC. (JP) 2006-10-31 US disclosed
CN-1708502-A Cephem compounds FUJISAWA PHARMACEUTICAL CO (JP) 2005-12-14 CN disclosed
EP-1556389-A1 CEPHEM COMPOUNDS Astellas Pharma Inc. (JP) 2005-07-27 EP disclosed
US-20040132994-A1 Cephem compounds FUJISAWA PHARMACEUTICAL CO., LTD (JP) 2004-07-08 US disclosed
WO-2004039814-A1 CEPHEM COMPOUNDS ASTELLAS PHARMA INC. (JP) 2004-05-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070037786-A1 Cephem compounds CEP170, ABCB11, SLC7A1 BRD9 3009/4885KAT2B 328/4885BRD4 3535/4885
US-20040132994-A1 Cephem compounds CEP170, ABCB11, RCC2 BRD9 2975/4885KAT2B 488/4885BRD4 3504/4885
US-20090012054-A1 Cephem Compounds and Use as Antimicrobial Agents CEP170, Q6ZSR9, H1-10 BRD9 790/4885KAT2B 712/4885BRD4 863/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.