SCHEMBL6070495

SCHEMBL6070495

CCCC1CCN(CCOc2cccc(-c3noc4ccsc34)c2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 3/20 0.40
HTR1A P08908 2/20 0.40
DRD2 P14416 1/20 0.40
HTR6 P50406 1/20 0.40
LTA4H P09960 1/20 0.40
BACE1 P56817 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
GPR119 Q8TDV5 1/20 0.38
KDM4E B2RXH2 2/20 0.38
HRH3 Q9Y5N1 4/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
MAOB P27338 1/20 0.37
KCNH2 Q12809 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6070752 0.89 HRH3 (0.47) LTA4HBACE1MEN1KMT2AKDM4E
SCHEMBL6069752 0.86 LTA4H (0.55) LTA4HBACE1KDM4EHRH3SMN1; SMN2
SCHEMBL6070257 0.85 BACE1 (0.56) LTA4HBACE1KDM4EHRH3SMN1; SMN2
SCHEMBL6069522 0.85 BACE1 (0.56) LTA4HBACE1KDM4EHRH3SMN1; SMN2
SCHEMBL1377022 0.85 BACE1 (0.56) LTA4HBACE1KDM4EHRH3SMN1; SMN2
SCHEMBL6070196 0.85 LTA4H (0.45) HTR7HTR1ALTA4HBACE1HRH3
Hydrochloric Acid SCHEMBL6069894 0.84 LTA4H (0.44) HTR7HTR1ALTA4HBACE1MEN1
SCHEMBL1377237 0.81 LTA4H (0.47) HTR7HTR1ADRD2LTA4HBACE1
SCHEMBL1376907 0.80 HTR7 (0.40) HTR7HTR1ADRD2HTR6LTA4H
SCHEMBL6070692 0.80 HRH3 (0.52) LTA4HBACE1KDM4EHRH3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7091199-B1 Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists AVENTIS PHARMACEUTICALS INC. (US) 2006-08-15 US claimed
EP-1216249-B1 THIENOISOXAZOLE PHENOXY UNSUBSTITUTED ETHYL AND PROPYL DERIVATIVES USEFUL AS D4 ANTAGONISTS AVENTIS PHARMA INC (US) 2003-11-19 EP claimed
US-7091199-B1 Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists AVENTIS PHARMACEUTICALS INC. (US) 2006-08-15 US disclosed
EP-1216249-B1 THIENOISOXAZOLE PHENOXY UNSUBSTITUTED ETHYL AND PROPYL DERIVATIVES USEFUL AS D4 ANTAGONISTS AVENTIS PHARMA INC (US) 2003-11-19 EP disclosed