SCHEMBL6072849

SCHEMBL6072849

CCCCc1ccc(C(OC(=O)[C@H](N)CS)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.55
TRPV1 Q8NER1 1/20 0.42
ALDH1A1 P00352 2/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
S1PR2 O95136 2/20 0.39
S1PR1 P21453 2/20 0.39
S1PR3 Q99500 1/20 0.38
RARB P10826 1/20 0.38
PLK1 P53350 1/20 0.38
SPHK1 Q9NYA1 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL232514 0.84 KIF11 (0.42) KIF11
Butylbenzyl SCHEMBL28861807 0.76 KIF11 (0.56) KIF11TRPV1ALDH1A1HPGDHSD17B10
SCHEMBL11106023 0.73 KIF11 (0.48) KIF11TRPV1ALDH1A1HPGDHSD17B10
SCHEMBL3318601 0.73 KIF11 (0.48) KIF11
SCHEMBL11199017 0.72 SPHK1 (0.50) ALDH1A1S1PR2S1PR1S1PR3SPHK1
SCHEMBL1899105 0.72 KIF11 (0.44) KIF11
SCHEMBL8636658 0.70 MMP2 (0.38) KIF11ALDH1A1
SCHEMBL7486608 0.70 KIF11 (0.42) KIF11
SCHEMBL7486605 0.70 KIF11 (0.42) KIF11
SCHEMBL2640404 0.69 PRSS1 (0.43) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006024453-A1 PYRAZOLOPYRIMIDINONES AS PHOSPHODIESTERASE INHIBITORS CTG PHARMA S.R.L. (IT) 2006-03-09 WO disclosed