SCHEMBL6072910

SCHEMBL6072910

CC(C)Oc1cc(F)ccc1N1CCN(CCCN2C(=O)CSC2=O)CC1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 15/20 0.51
ADRA1B P35368 14/20 0.51
ADRA1D P25100 11/20 0.51
HTR1A P08908 2/20 0.44
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTR7 P34969 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6072693 0.99 ADRA1A (0.51) ADRA1AADRA1BADRA1DHTR1AMEN1
SCHEMBL6072722 0.98 ADRA1B (0.51) ADRA1AADRA1BADRA1DHTR1AMEN1
Hydrochloric Acid SCHEMBL6072738 0.97 ADRA1B (0.51) ADRA1AADRA1BADRA1DHTR1AMEN1
SCHEMBL6073161 0.92 ADRA1A (0.44) ADRA1AADRA1BADRA1DHTR1AMEN1
Hydrochloric Acid SCHEMBL6072912 0.91 ADRA1B (0.43) ADRA1AADRA1BADRA1DHTR1AMEN1
SCHEMBL6072742 0.90 ADRA1B (0.44) ADRA1AADRA1BADRA1DHTR1AMEN1
Hydrochloric Acid SCHEMBL6072701 0.89 ADRA1B (0.43) ADRA1AADRA1BADRA1DHTR1AMEN1
SCHEMBL6072734 0.89 ADRA1B (0.43) ADRA1AADRA1BADRA1DHTR1AMEN1
SCHEMBL6072696 0.89 HTR1A (0.53) ADRA1AADRA1BADRA1DHTR1AMEN1
Hydrochloric Acid SCHEMBL6073167 0.89 ADRA1B (0.43) ADRA1AADRA1BADRA1DHTR1AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006013445-A2 THIAZOLIDINEDIONE DERIVATIVES AS ALPHA ADRENERGIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2006-02-09 WO claimed
WO-2006013445-A2 THIAZOLIDINEDIONE DERIVATIVES AS ALPHA ADRENERGIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2006-02-09 WO disclosed