SCHEMBL6079183

SCHEMBL6079183

COC(=O)c1cc(NS(=O)(=O)c2ccc3ccc(NC(=S)Nc4ccc5ccc(S(=O)(=O)Nc6cccnc6)cc5c4)cc3c2)ccc1Cl

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.53
ALDH1A1 P00352 3/20 0.53
GAA P10253 2/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
TSHR P16473 1/20 0.47
MAPT P10636 4/20 0.46
IKBKB O14920 2/20 0.45
JAK2 O60674 2/20 0.45
ROCK2 O75116 2/20 0.45
JAK1 P23458 2/20 0.45
TYK2 P29597 2/20 0.45
JAK3 P52333 2/20 0.45
ROCK1 Q13464 2/20 0.45
STAT5A P42229 1/20 0.45
KMT2A Q03164 5/20 0.45
MEN1 O00255 4/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
CSF1R P07333 1/20 0.44
NAMPT P43490 2/20 0.43
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6079206 0.90 MEN1 (0.51) LMNAALDH1A1TSHRMAPTIKBKB
SCHEMBL6079143 0.90 ALDH1A1 (0.64) LMNAALDH1A1GAAL3MBTL1MAPT
SCHEMBL6078679 0.86 LMNA (0.56) LMNAALDH1A1GAAL3MBTL1MAPT
SCHEMBL6079922 0.86 MAPT (0.60) LMNAALDH1A1GAAL3MBTL1MAPT
SCHEMBL6078415 0.85 ALDH1A1 (0.59) LMNAALDH1A1GAAL3MBTL1TSHR
SCHEMBL6079074 0.85 LMNA (0.54) LMNAALDH1A1GAAL3MBTL1MAPT
SCHEMBL6078607 0.83 MEN1 (0.53) ALDH1A1TSHRIKBKBJAK2ROCK2
SCHEMBL6078277 0.82 LMNA (0.67) LMNAALDH1A1GAAL3MBTL1MAPT
SCHEMBL6079588 0.80 LMNA (0.49) LMNAALDH1A1GAAL3MBTL1MAPT
SCHEMBL6078676 0.80 LMNA (0.64) LMNAALDH1A1GAAL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7071231-B2 Naphthalene ureas as glucose uptake enhancers TELIK, INC. (US) 2006-07-04 US disclosed
US-6458998-B1 NAPHTHALENEUREAS AS ANTIDIABETIC AGENTS TELIK, INC. 2002-10-01 US disclosed