SCHEMBL6081377

SCHEMBL6081377

CC(C)C1CCCN1CCOc1ccc(-n2ccn(-c3ccc(Oc4ccccc4)cc3)c2=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 4/20 0.44
HRH3 Q9Y5N1 5/20 0.43
MCHR1 Q99705 5/20 0.43
KCNH2 Q12809 5/20 0.43
MCHR2 Q969V1 1/20 0.42
PTGER4 P35408 2/20 0.40
PTGER2 P43116 2/20 0.40
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1729474 0.87 HRH3 (0.57) HRH3KCNH2
SCHEMBL6081517 0.84 LTA4H (0.45) LTA4HHRH3MCHR1KCNH2MCHR2
SCHEMBL6081905 0.83 MCHR1 (0.48) LTA4HHRH3MCHR1KCNH2MCHR2
SCHEMBL6081914 0.83 MCHR1 (0.48) LTA4HHRH3MCHR1KCNH2MCHR2
SCHEMBL1727398 0.82 NPC1 (0.49) LTA4HHRH3MCHR1KCNH2MCHR2
SCHEMBL6081329 0.82 MCHR1 (0.49) LTA4HHRH3MCHR1KCNH2MCHR2
SCHEMBL1727509 0.81 LTA4H (0.42) LTA4HHRH3MCHR1KCNH2MCHR2
SCHEMBL6081581 0.81 LTA4H (0.50) LTA4HHRH3MCHR1KCNH2MCHR2
SCHEMBL6081488 0.80 MCHR1 (0.48) LTA4HHRH3MCHR1KCNH2MCHR2
SCHEMBL6081396 0.80 LTA4H (0.54) LTA4HHRH3MCHR1KCNH2PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7141561-B2 Substituted diaryl heterocycles, process for their preparation and their use as medicaments SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-11-28 US disclosed