SCHEMBL6091353

SCHEMBL6091353

Cc1[nH]c(C=O)c(C)c1CN1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.45
KMT2A Q03164 7/20 0.42
MEN1 O00255 6/20 0.42
HSD17B10 Q99714 5/20 0.42
ALDH1A1 P00352 7/20 0.40
KDM4E B2RXH2 6/20 0.40
POLB P06746 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HPGD P15428 2/20 0.39
MAPT P10636 5/20 0.38
CHRNA7 P36544 1/20 0.38
CASP1 P29466 2/20 0.36
CFB P00751 1/20 0.35
ERN1 O75460 1/20 0.35
TSHR P16473 1/20 0.34
ERAP1 Q9NZ08 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6092642 0.98 ALOX15 (0.42) ALOX15KMT2AMEN1HSD17B10ALDH1A1
SCHEMBL6089632 0.84 HSD17B10 (0.44) KMT2AMEN1HSD17B10ALDH1A1KDM4E
SCHEMBL7125283 0.84 PDGFRB (0.34) ALOX15KMT2AMEN1HSD17B10ALDH1A1
SCHEMBL5401530 0.83 MCL1 (0.40) KMT2AMEN1HSD17B10ALDH1A1KDM4E
SCHEMBL7117376 0.83 ALDH1A1 (0.34) KMT2AMEN1HSD17B10ALDH1A1KDM4E
SCHEMBL6089855 0.83 HRH3 (0.42) ALOX15KMT2AMEN1ALDH1A1POLB
SCHEMBL7125898 0.82 ALDH1A1 (0.43) HSD17B10ALDH1A1KDM4EPOLBHPGD
SCHEMBL6092029 0.81 PDGFRB (0.46) ALOX15KMT2AL3MBTL1MAPT
SCHEMBL7117883 0.81 HRH3 (0.42) KMT2AMEN1ALDH1A1KDM4EL3MBTL1
SCHEMBL7128643 0.81 TRPV6 (0.35) KMT2AMEN1HSD17B10ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed
EP-1218373-A2 2-PYRAZOLIN-5-ONES AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2002-07-03 EP disclosed
WO-2001009121-A2 2-PYRAZOLIN-5-ONES_AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-02-08 WO disclosed