SCHEMBL6092765

SCHEMBL6092765

CCOC(=O)C(C)(C)Oc1ccc(-c2cccs2)cc1CBr

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 6/20 0.46
HDAC2 Q92769 6/20 0.46
HDAC3 O15379 5/20 0.46
FBP1 P09467 7/20 0.42
ABCB11 O95342 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
HTR2A P28223 1/20 0.39
PMP22 Q01453 1/20 0.39
PPARA Q07869 1/20 0.39
KCNH2 Q12809 1/20 0.39
KMT2A Q03164 1/20 0.38
TNFRSF1A P19438 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6094551 0.90 HDAC1 (0.47) HDAC1HDAC2HDAC3FBP1ABCB11
SCHEMBL6094343 0.82 ERN1 (0.50) HDAC1HDAC2HDAC3FBP1TNFRSF1A
SCHEMBL6094560 0.82 TNFRSF1A (0.48) HDAC1HDAC2HDAC3FBP1KMT2A
SCHEMBL6092109 0.81 ALDH1A1 (0.41) HDAC1HDAC2HDAC3FBP1ABCB11
SCHEMBL14110370 0.80 FBP1 (0.49) FBP1ABCB11CYP1A2CYP3A4TSHR
SCHEMBL4685610 0.77 FBP1 (0.53) FBP1ABCB11CYP1A2CYP3A4TSHR
SCHEMBL6091552 0.76 ALDH1A1 (0.41) HDAC1HDAC2HDAC3FBP1ABCB11
SCHEMBL6093858 0.75 ALDH1A1 (0.47) KCNH2KMT2ATNFRSF1A
SCHEMBL6092795 0.75 FBP1 (0.46) HDAC1HDAC2HDAC3FBP1ABCB11
SCHEMBL6091509 0.74 TNFRSF1A (0.37) HDAC1HDAC2HDAC3TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060063828-A1 1,2-Bis-(substituted-phenyl)-2-propen-1-ones and pharmaceutical compositions thereof ATHEROGENICS, INC. 2006-03-23 US disclosed
WO-2006004903-A2 1,2-BIS-(SUBSTITUTED-PHENYL)-2-PROPEN-1-ONES AND PHARMACEUTICAL COMPOSITIONS THEREOF ATHEROGENICS, INC. (US) 2006-01-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060063828-A1 1,2-Bis-(substituted-phenyl)-2-propen-1-ones and pharmaceutical compositions thereof ABCB11, CEL, CYP46A1 HDAC1 1097/4885HDAC2 651/4885HDAC3 735/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.