SCHEMBL6109302

SCHEMBL6109302

O=C(O)N(C(=O)Oc1ccccc1)c1cc(Oc2ccc3c(ccn3C(=O)NC3CC3)c2)ccn1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 3/20 0.37
KDR P35968 10/20 0.36
NPC1 O15118 1/20 0.35
RET P07949 1/20 0.34
PDGFRA P16234 1/20 0.34
ABL1 P00519 1/20 0.34
TNKS O95271 1/20 0.33
DGAT1 O75907 1/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5102304 0.97 RIPK1 (0.38) RIPK1KDRNPC1RETPDGFRA
SCHEMBL5101380 0.93 KDR (0.39) RIPK1KDRDGAT1RAB9A
SCHEMBL6375561 0.85 KDR (0.35) KDR
SCHEMBL1893391 0.85 KDR (0.39) KDRRETPDGFRA
SCHEMBL5113619 0.84 GCK (0.40) KDR
SCHEMBL1899097 0.84 KDR (0.38) KDRRETPDGFRA
SCHEMBL6038526 0.83 RAB9A (0.38) KDRNPC1HPGDRAB9A
SCHEMBL5107702 0.82 GCK (0.42) RIPK1KDRABL1
SCHEMBL5101397 0.82 KDR (0.36) KDR
SCHEMBL6038768 0.82 SMN1; SMN2 (0.38) KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7109219-B2 Nitrogen-containing aromatic derivatives EISAI CO., LTD. (JP) 2006-09-19 US disclosed