SCHEMBL6111192

SCHEMBL6111192

COc1ccccc1-c1nc(C)c(C#N)c(S)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.52
KDM4E B2RXH2 8/20 0.52
HPGD P15428 4/20 0.52
SQOR Q9Y6N5 1/20 0.47
ADORA2A P29274 1/20 0.46
ADORA1 P30542 1/20 0.46
HSD17B10 Q99714 4/20 0.45
TSHR P16473 3/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
BLM P54132 1/20 0.44
HTT P42858 2/20 0.43
NPSR1 Q6W5P4 2/20 0.41
LMNA P02545 3/20 0.40
L3MBTL1 Q9Y468 3/20 0.40
MAPT P10636 2/20 0.40
ATM Q13315 1/20 0.40
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
CYP1A2 P05177 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6110675 0.83 CRHR1 (0.47) ALDH1A1KDM4EADORA2AADORA1HSD17B10
SCHEMBL6110296 0.80 KDM4E (0.38) ALDH1A1KDM4EHPGDADORA2AADORA1
SCHEMBL5809944 0.76 PDE4B (0.51) ALDH1A1KDM4EHPGDSQORADORA2A
SCHEMBL6112336 0.73 ADORA2A (0.50) ALDH1A1KDM4EHPGDSQORADORA2A
SCHEMBL23066466 0.73 ALDH1A1 (0.61) ALDH1A1KDM4EHPGDHSD17B10TSHR
SCHEMBL17971412 0.70 ALDH1A1 (0.52) ALDH1A1KDM4EHPGDSQORADORA2A
SCHEMBL6253695 0.69 KDM4E (1.00) ALDH1A1KDM4EHPGDADORA2AADORA1
SCHEMBL6109551 0.68 KDM4E (0.51) ALDH1A1KDM4EHPGDADORA2AADORA1
SCHEMBL14983662 0.67 CYP1A2 (0.51) ALDH1A1KDM4EHPGDHSD17B10TSHR
SCHEMBL8802694 0.66 KDM4E (0.48) ALDH1A1KDM4EHPGDSQORADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006010568-A2 SUBSTITUTED PYRIDO[3',2':4,5]THIENO[3,2-D]PYRIMIDINE-2,4(1 H,3H)-DIONES AND -4(3H)-ONES, PYRIDO[3',2':4,5]FURO[3,2-D]PYRIMIDINE-2,4(1 H,3H)-DIONES AND -4(3H)-ONES, AND USE THEREOF AS INHIBITORS OF TNF-ALPHA RELEASE CURACYTE DISCOVERY GMBH (DE) 2006-02-02 WO disclosed