SCHEMBL5809944

SCHEMBL5809944

Cc1nc(-c2ccccc2)nc(S)c1C#N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.51
PDE4D Q08499 1/20 0.51
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
ADORA2A P29274 6/20 0.47
ADORA1 P30542 6/20 0.47
HSD17B10 Q99714 3/20 0.47
HPGD P15428 4/20 0.45
ALDH1A1 P00352 3/20 0.45
HTT P42858 2/20 0.45
KDM4E B2RXH2 2/20 0.45
ADRA2A P08913 1/20 0.45
LMNA P02545 1/20 0.45
SQOR Q9Y6N5 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
ADORA2B P29275 1/20 0.43
NPSR1 Q6W5P4 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6109551 0.83 KDM4E (0.51) MEN1KMT2AADORA2AADORA1HSD17B10
SCHEMBL5805731 0.80 LMNA (0.62) PDE4BPDE4DMEN1KMT2AADORA2A
SCHEMBL6112336 0.80 ADORA2A (0.50) MEN1KMT2AADORA2AADORA1HPGD
SCHEMBL6110296 0.78 KDM4E (0.38) PDE4BPDE4DKMT2AADORA2AADORA1
SCHEMBL1321790 0.78 NPSR1 (0.37) PDE4BPDE4DMEN1KMT2AADORA2A
SCHEMBL6111192 0.76 ALDH1A1 (0.52) MEN1KMT2AADORA2AADORA1HSD17B10
SCHEMBL5809819 0.75 L3MBTL1 (0.44) MEN1KMT2AADORA2AADORA1HSD17B10
SCHEMBL27429230 0.73 ADORA1 (0.60) PDE4BPDE4DMEN1KMT2AADORA2A
SCHEMBL1320853 0.72 L3MBTL1 (0.68) MEN1KMT2AADORA2AADORA1HSD17B10
SCHEMBL19313821 0.71 ADORA1 (0.52) MEN1KMT2AADORA2AADORA1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006100095-A1 SUBSTITUTED CARBOXAMIDES METHOD FOR PRODUCTION AND USE THEREOF AS TNF-ALPHA RELEASE INHIBITORS CURACYTE DISCOVERY GMBH (DE) 2006-09-28 WO disclosed