SCHEMBL6127410

SCHEMBL6127410

[NH]c1ccc([C@@H]2CC[C@@H](c3ccc([NH])cc3)N2c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.42
HTR2C P28335 3/20 0.40
PRKCZ Q05513 2/20 0.40
CA12 O43570 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
DEGS1 O15121 1/20 0.36
CYP3A4 P08684 2/20 0.36
SLC6A9 P48067 1/20 0.36
BCHE P06276 1/20 0.34
ACHE P22303 1/20 0.34
HRH4 Q9H3N8 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1982165 0.84 KIF11 (0.47) NOTUMHTR2CPRKCZCA12CA2
SCHEMBL1982310 0.84 CYP3A4 (0.41) NOTUMHTR2CPRKCZCA12CA2
SCHEMBL1983109 0.84 CYP3A4 (0.41) NOTUMHTR2CPRKCZCA12CA2
SCHEMBL6123402 0.84 CYP3A4 (0.41) NOTUMHTR2CPRKCZCA12CA2
SCHEMBL1983143 0.84 KIF11 (0.47) NOTUMHTR2CPRKCZCA12CA2
SCHEMBL1988497 0.84 CYP3A4 (0.41) NOTUMHTR2CPRKCZCA12CA2
SCHEMBL2374410 0.84 RIPK1 (0.38) PRKCZCYP3A4ACHEHRH3
SCHEMBL1989822 0.84 RIPK1 (0.38) PRKCZCYP3A4ACHEHRH3
SCHEMBL1985242 0.74 LPL (0.38) NOTUMHTR2CPRKCZCA2CA9
SCHEMBL1985257 0.74 LPL (0.38) NOTUMHTR2CPRKCZCA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2455376-A1 Heterocyclic compounds as inhibitors of hepatitis C virus (HCV) Abbott Laboratories (US) 2012-05-23 EP disclosed