SCHEMBL6131646

SCHEMBL6131646

CC(C)(C)c1ccc(Nc2ccc(-c3ccc(Nc4ccc(C(C)(C)C)cc4)c(-c4ccc(Br)cc4)c3)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.39
AKR1C2 P52895 3/20 0.39
KIF11 P52732 3/20 0.38
XDH P47989 1/20 0.37
SLC22A12 Q96S37 1/20 0.37
APP P05067 1/20 0.35
CNR1 P21554 1/20 0.35
ACP1 P24666 1/20 0.35
SLC2A1 P11166 1/20 0.34
MAPKAPK2 P49137 1/20 0.34
RAPGEF4 Q8WZA2 1/20 0.34
THRB P10828 1/20 0.33
TGFBR1 P36897 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31013582 0.91 AKR1C3 (0.44) AKR1C3AKR1C2KIF11XDHSLC22A12
SCHEMBL31013592 0.85 HSD17B2 (0.44) AKR1C3AKR1C2KIF11XDHSLC22A12
SCHEMBL31013596 0.85 HSD17B2 (0.44) AKR1C3AKR1C2KIF11XDHSLC22A12
SCHEMBL1086771 0.84 RAPGEF4 (0.50) AKR1C3AKR1C2APPACP1MAPKAPK2
SCHEMBL10002566 0.84 RAPGEF4 (0.44) AKR1C3AKR1C2APPMAPKAPK2RAPGEF4
SCHEMBL24175562 0.83 AKR1C3 (0.46) AKR1C3AKR1C2KIF11XDHSLC22A12
SCHEMBL4629998 0.82 AKR1C3 (0.36) AKR1C3AKR1C2KIF11XDHSLC22A12
SCHEMBL6131645 0.81 APP (0.48) AKR1C3AKR1C2KIF11XDHSLC22A12
SCHEMBL4629995 0.81 APP (0.48) AKR1C3AKR1C2KIF11XDHSLC22A12
SCHEMBL30675131 0.80 ALDH1A1 (0.50) AKR1C3AKR1C2ACP1MAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6956095-B2 Process for producing aryl—aryl coupled compounds COVION ORGANIC SEMICONDUCTORS GMBH (DE) 2005-10-18 US disclosed