SCHEMBL6131821

SCHEMBL6131821

COc1cc(CN2CCN(c3ccccn3)CC2)c(Br)cc1OCc1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.71
HTT P42858 4/20 0.71
KDM4E B2RXH2 4/20 0.71
LMNA P02545 4/20 0.71
MAPK1 P28482 3/20 0.71
TSHR P16473 2/20 0.71
SMN1; SMN2 Q16637 2/20 0.57
HPGD P15428 1/20 0.57
ALOX12 P18054 1/20 0.57
RAB9A P51151 3/20 0.56
NPC1 O15118 2/20 0.56
MAPT P10636 2/20 0.56
EHMT2 Q96KQ7 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
HSD17B10 Q99714 2/20 0.48
HTR1A P08908 2/20 0.48
ADRA1D P25100 1/20 0.48
ADRA1A P35348 1/20 0.48
ADRA1B P35368 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6131842 0.98 ALDH1A1 (0.69) ALDH1A1HTTKDM4ELMNAMAPK1
SCHEMBL6131898 0.88 ALDH1A1 (0.71) ALDH1A1HTTKDM4ELMNAMAPK1
SCHEMBL6131919 0.86 ALDH1A1 (0.69) ALDH1A1HTTKDM4ELMNAMAPK1
SCHEMBL4750766 0.83 ALDH1A1 (0.92) ALDH1A1HTTKDM4ELMNAMAPK1
SCHEMBL6131770 0.83 ALDH1A1 (0.56) ALDH1A1HTTKDM4ELMNAMAPK1
SCHEMBL6131961 0.83 DRD2 (0.58) ALDH1A1HTTKDM4ELMNAMAPK1
SCHEMBL6131838 0.82 DRD2 (0.56) ALDH1A1HTTKDM4ELMNAMAPK1
SCHEMBL7686968 0.81 ALDH1A1 (0.54) ALDH1A1HTTKDM4ELMNAMAPK1
Bicarbonate SCHEMBL6131884 0.80 ALDH1A1 (0.51) ALDH1A1HTTKDM4ELMNAMAPK1
Bicarbonate SCHEMBL6131829 0.80 ALDH1A1 (0.51) ALDH1A1HTTKDM4ELMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP claimed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP claimed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO claimed
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP disclosed
US-6479495-B1 SIMULTANEOUSLY TREATING DEPRESSION AND MEMORY DYSFUNCTION IN MAMMALS SUFFERING FROM MEMORY DYSFUNCTION AND DEPRESSION AVENTIS PHARMACEUTICALS INC. 2002-11-12 US disclosed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP disclosed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO disclosed