Bicarbonate

Bicarbonate

SCHEMBL6131829

COc1cc(CN2CCN(c3ccccn3)CC2)c(Br)cc1OC(=O)N(C)C.COc1cc(CN2CCN(c3ccccn3)CC2)c(Br)cc1OC(=O)N(C)C.O=C([O-])[O-].[Cs+].[Cs+]

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.51
KDM4E B2RXH2 8/20 0.51
SMN1; SMN2 Q16637 3/20 0.47
DRD3 P35462 1/20 0.47
LMNA P02545 3/20 0.47
TSHR P16473 3/20 0.47
MAPK1 P28482 2/20 0.47
HTT P42858 2/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
HSD17B10 Q99714 5/20 0.45
HPGD P15428 2/20 0.45
MAPT P10636 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
TP53 P04637 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL6131884 1.00 ALDH1A1 (0.51) ALDH1A1KDM4ESMN1; SMN2DRD3LMNA
SCHEMBL7686968 0.96 ALDH1A1 (0.54) ALDH1A1KDM4ESMN1; SMN2DRD3LMNA
SCHEMBL6131859 0.86 ALDH1A1 (0.54) ALDH1A1KDM4ESMN1; SMN2LMNATSHR
SCHEMBL6131848 0.86 ALDH1A1 (0.54) ALDH1A1KDM4ESMN1; SMN2LMNATSHR
SCHEMBL6131963 0.82 KDM4E (0.60) ALDH1A1KDM4ESMN1; SMN2DRD3LMNA
SCHEMBL6132095 0.81 ALDH1A1 (0.64) ALDH1A1KDM4ESMN1; SMN2LMNATSHR
SCHEMBL6131812 0.81 ALDH1A1 (0.52) ALDH1A1KDM4ESMN1; SMN2DRD3LMNA
SCHEMBL6131821 0.80 ALDH1A1 (0.71) ALDH1A1KDM4ESMN1; SMN2LMNATSHR
SCHEMBL6131961 0.79 DRD2 (0.58) ALDH1A1KDM4ESMN1; SMN2DRD3LMNA
SCHEMBL6131770 0.79 ALDH1A1 (0.56) ALDH1A1KDM4ESMN1; SMN2DRD3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP disclosed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP disclosed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO disclosed