SCHEMBL6131865

SCHEMBL6131865

COc1cc(CCN2CCN(c3ccc4ccccc4n3)CC2)ccc1OC(C)=O

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
DRD3 P35462 3/20 0.48
ABCB1 P08183 1/20 0.48
ADRA1D P25100 2/20 0.48
ADRA1A P35348 2/20 0.48
ADRA1B P35368 2/20 0.48
PKM P14618 1/20 0.48
EBP Q15125 2/20 0.47
SIGMAR1 Q99720 2/20 0.47
TMEM97 Q5BJF2 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
DRD2 P14416 2/20 0.47
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
NOD2 Q9HC29 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6131988 0.90 DRD3 (0.48) NPC1RAB9ADRD3ABCB1ADRA1D
SCHEMBL6131991 0.90 DRD3 (0.48) NPC1RAB9ADRD3ABCB1ADRA1D
SCHEMBL6131974 0.85 NPC1 (0.54) NPC1RAB9ADRD3ADRA1DADRA1A
SCHEMBL6131794 0.81 ADRA1D (0.68) ADRA1DADRA1AADRA1BDRD2
SCHEMBL6131869 0.79 ADRA1D (0.60) DRD3ADRA1DADRA1AADRA1BEBP
SCHEMBL6131937 0.79 ADRA1D (0.60) ADRA1DADRA1AADRA1BEBPSIGMAR1
SCHEMBL6131777 0.79 ADRA1D (0.59) ADRA1DADRA1AADRA1BEBPSIGMAR1
SCHEMBL6131863 0.78 HRH3 (0.51) NPC1RAB9AHRH3KMT2A
SCHEMBL6131802 0.77 ADRA1D (0.81) ADRA1DADRA1AADRA1BKMT2A
SCHEMBL6131819 0.76 ADRA1D (0.56) ADRA1DADRA1AADRA1BEBPSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP disclosed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP disclosed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO disclosed