SCHEMBL6131988

SCHEMBL6131988

COc1cc(CCN2CCN(c3ccc4ccccc4n3)CC2)ccc1OC(=O)N(C)C

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 3/20 0.48
ABCB1 P08183 1/20 0.48
PKM P14618 1/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
NOD2 Q9HC29 1/20 0.46
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
EBP Q15125 2/20 0.45
SIGMAR1 Q99720 2/20 0.45
DRD2 P14416 2/20 0.45
TMEM97 Q5BJF2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6131865 0.90 NPC1 (0.49) DRD3ABCB1PKMNPC1RAB9A
SCHEMBL6131991 0.89 DRD3 (0.48) DRD3ABCB1PKMNPC1RAB9A
SCHEMBL6131908 0.84 ALDH1A1 (0.58) DRD3NPC1RAB9AMEN1KMT2A
Hydrochloric Acid SCHEMBL6132036 0.84 ALDH1A1 (0.57) DRD3NPC1RAB9AMEN1KMT2A
SCHEMBL6131974 0.83 NPC1 (0.54) DRD3NPC1RAB9AKMT2AADRA1D
SCHEMBL6131790 0.81 ADRA1D (0.57) DRD3MEN1KMT2AADRA1DADRA1A
SCHEMBL6131925 0.81 ADRA1D (0.57) KMT2AADRA1DADRA1AADRA1BEBP
Hydrochloric Acid SCHEMBL6131948 0.78 ADRA1D (0.54) KMT2AADRA1DADRA1AADRA1BSIGMAR1
SCHEMBL6131889 0.78 ADRA1D (0.76) KMT2AADRA1DADRA1AADRA1B
SCHEMBL6131931 0.78 ADRA1D (0.53) ADRA1DADRA1AADRA1BEBPSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP claimed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP claimed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO claimed