SCHEMBL6131937

SCHEMBL6131937

COc1cc(CCN2CCN(c3ccccc3C)CC2)ccc1OC(C)=O

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 4/20 0.60
ADRA1A P35348 4/20 0.60
ADRA1B P35368 4/20 0.60
ALDH1A1 P00352 2/20 0.52
TSHR P16473 2/20 0.52
KMT2A Q03164 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
EBP Q15125 2/20 0.52
SIGMAR1 Q99720 2/20 0.52
TMEM97 Q5BJF2 1/20 0.52
HTR1A P08908 4/20 0.52
KDM4E B2RXH2 1/20 0.52
ALOX15 P16050 1/20 0.52
HTR1D P28221 1/20 0.51
HTR1B P28222 1/20 0.51
HTR2C P28335 2/20 0.50
DRD2 P14416 1/20 0.50
DRD1 P21728 1/20 0.50
HTR2A P28223 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6131794 0.92 ADRA1D (0.68) ADRA1DADRA1AADRA1BHTR1AHTR2C
SCHEMBL6131869 0.90 ADRA1D (0.60) ADRA1DADRA1AADRA1BKMT2AEBP
SCHEMBL6131928 0.89 ADRA1D (0.57) ADRA1DADRA1AADRA1BALDH1A1TSHR
SCHEMBL6131925 0.89 ADRA1D (0.57) ADRA1DADRA1AADRA1BALDH1A1TSHR
SCHEMBL6131777 0.89 ADRA1D (0.59) ADRA1DADRA1AADRA1BALDH1A1EBP
Hydrochloric Acid SCHEMBL6132049 0.87 ADRA1D (0.55) ADRA1DADRA1AADRA1BALDH1A1TSHR
SCHEMBL6131802 0.87 ADRA1D (0.81) ADRA1DADRA1AADRA1BALDH1A1KMT2A
SCHEMBL6131819 0.86 ADRA1D (0.56) ADRA1DADRA1AADRA1BEBPSIGMAR1
SCHEMBL6131986 0.84 LMNA (0.60) ADRA1DADRA1AADRA1BALDH1A1NPSR1
SCHEMBL6131865 0.79 NPC1 (0.49) ADRA1DADRA1AADRA1BKMT2AEBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP disclosed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP disclosed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO disclosed