SCHEMBL6135722

SCHEMBL6135722

Nc1ccccc1CC1(C(=O)O)CCN(C(=O)O)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.37
AGTR2 P50052 2/20 0.35
OPRK1 P41145 1/20 0.34
KMT2A Q03164 2/20 0.34
SIGMAR1 Q99720 1/20 0.34
TET3 O43151 1/20 0.34
FBXL19 Q6PCT2 1/20 0.34
CXXC5 Q7LFL8 1/20 0.34
TET1 Q8NFU7 1/20 0.34
KDM2B Q8NHM5 1/20 0.34
CXXC4 Q9H2H0 1/20 0.34
KDM2A Q9Y2K7 1/20 0.34
ALDH1A1 P00352 3/20 0.34
RAB9A P51151 3/20 0.34
NPC1 O15118 2/20 0.33
MEN1 O00255 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP2D6 P10635 1/20 0.33
CPB2 Q96IY4 1/20 0.33
RIPK1 Q13546 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3485621 0.80 AVPR1A (0.44) OPRM1KMT2AALDH1A1RAB9ANPC1
SCHEMBL28761351 0.79 SLC6A2 (0.39) OPRM1CYP2D6
SCHEMBL27644978 0.79 RAB9A (0.44) SIGMAR1ALDH1A1RAB9A
SCHEMBL2463164 0.75 NAAA (0.44) ALDH1A1MAPK1CYP2D6
SCHEMBL17870745 0.72 CYP2C19 (0.37) OPRM1OPRK1KMT2ASIGMAR1ALDH1A1
SCHEMBL1177807 0.72 ESR1 (0.41) OPRK1ALDH1A1RAB9ANPC1
SCHEMBL10006856 0.72 P2RX7 (0.36) ALDH1A1RAB9ANPC1
SCHEMBL2468103 0.71 PLA2G10 (0.41) KMT2AALDH1A1MEN1
SCHEMBL28250538 0.71 RAB9A (0.43) SIGMAR1ALDH1A1RAB9A
SCHEMBL3984421 0.71 KMT2A (0.46) KMT2ATET3FBXL19CXXC5KDM2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100558428-C Calcitonin gene related peptide receptor antagonists BRISTOL MYERS SQUIBB CO (US) 2009-11-11 CN disclosed
CN-1917921-A Calcitonin gene related peptide receptor antagonists BRISTOL MYERS SQUIBB CO (US) 2007-02-21 CN disclosed
EP-1539766-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS Bristol-Myers Squibb Company (US) 2005-06-15 EP disclosed
WO-2003104236-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-12-18 WO disclosed