SCHEMBL6137426

SCHEMBL6137426

NC(N)=NC(=O)c1ccc(N2CCN(C(=O)c3ccc(F)cc3)CC2)c(C(F)(F)F)c1

nearest known ligand 0.71

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 20/20 0.71
CYP2C19 P33261 6/20 0.71
CYP3A4 P08684 6/20 0.71
CYP2C9 P11712 7/20 0.69
CYP2D6 P10635 2/20 0.60
KCNH2 Q12809 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7985442 0.84 SLC9A1 (0.53) SLC9A1CYP2C19CYP3A4CYP2C9CYP2D6
SCHEMBL6137546 0.84 SLC9A1 (0.53) SLC9A1CYP2C19CYP3A4CYP2C9CYP2D6
Sabiporide SCHEMBL1286663 0.83 SLC9A1 (1.00) SLC9A1CYP2C19CYP3A4CYP2C9CYP2D6
Sabiporide SCHEMBL1286649 0.83 SLC9A1 (0.98) SLC9A1CYP2C19CYP3A4CYP2C9CYP2D6
Sabiporide SCHEMBL4901735 0.82 SLC9A1 (0.96) SLC9A1CYP2C19CYP3A4CYP2C9CYP2D6
SCHEMBL6137414 0.81 SLC9A1 (0.48) SLC9A1CYP2C19CYP3A4CYP2C9
SCHEMBL7985451 0.80 ALDH1A1 (0.54) SLC9A1CYP2C19CYP3A4
Sabiporide SCHEMBL27472449 0.79 SLC9A1 (0.89) SLC9A1CYP2C19CYP3A4CYP2C9CYP2D6
Hydrochloric Acid SCHEMBL7837958 0.79 SLC9A1 (0.62) SLC9A1CYP2C19CYP3A4CYP2C9CYP2D6
SCHEMBL7985439 0.77 NPY2R (0.46) SLC9A1CYP2C19CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165534-B1 BENZOYLGUANIDINE DERIVATIVES WITH ADVANTAGEOUS PROPERTIES, METHOD FOR PRODUCING THEM AND THEIR USE IN THE PRODUCTION OF MEDICAMENTS BOEHRINGER INGELHEIM PHARMA (DE) 2005-02-02 EP claimed