SCHEMBL6139039

SCHEMBL6139039

COCC1CCCN1NS(=O)(=O)c1c(Cl)ccc([N+](=O)[O-])c1Cl

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 6/20 0.35
CASP7 P55210 5/20 0.35
CASP9 P55211 1/20 0.35
VCAM1 P19320 3/20 0.35
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
MCOLN3 Q8TDD5 1/20 0.34
LMNA P02545 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
NPBWR1 P48145 1/20 0.34
MCHR1 Q99705 1/20 0.34
HDAC8 Q9BY41 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
HDAC1 Q13547 1/20 0.34
KCNH2 Q12809 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2769590 1.00 CASP3 (0.35) CASP3CASP7CASP9VCAM1ALDH1A1
SCHEMBL2768975 1.00 CASP3 (0.35) CASP3CASP7CASP9VCAM1ALDH1A1
SCHEMBL2768514 0.90 VCAM1 (0.36) CASP3CASP7CASP9VCAM1ALDH1A1
SCHEMBL2768872 0.90 VCAM1 (0.36) CASP3CASP7CASP9VCAM1ALDH1A1
SCHEMBL6137742 0.90 VCAM1 (0.36) CASP3CASP7CASP9VCAM1ALDH1A1
SCHEMBL6563969 0.83 CASP3 (0.46) CASP3CASP7CASP9ALDH1A1KMT2A
SCHEMBL2767458 0.78 HDAC8 (0.37) CASP3CASP7CASP9HDAC8HDAC6
SCHEMBL2769019 0.78 HDAC8 (0.37) CASP3CASP7CASP9HDAC8HDAC6
SCHEMBL6138091 0.78 HDAC8 (0.37) CASP3CASP7CASP9HDAC8HDAC6
SCHEMBL6564147 0.76 CASP3 (0.45) CASP3CASP7CASP9ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1272175-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2005-08-31 EP disclosed
EP-1272175-A2 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2003-01-08 EP disclosed
WO-2001072960-A2 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2001-10-04 WO disclosed