SCHEMBL6137742

SCHEMBL6137742

COCC1CCCN1NS(=O)(=O)c1c(Cl)ccc([N+](=O)[O-])c1O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 2/20 0.36
CASP3 P42574 5/20 0.35
CASP7 P55210 4/20 0.35
NPBWR1 P48145 1/20 0.35
MCHR1 Q99705 1/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HDAC1 Q13547 1/20 0.35
CASP9 P55211 1/20 0.34
KMT2A Q03164 3/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP2D6 P10635 1/20 0.34
MAPT P10636 1/20 0.34
MEN1 O00255 1/20 0.34
HPGD P15428 1/20 0.34
TXNRD1 Q16881 1/20 0.33
SCN9A Q15858 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2768872 1.00 VCAM1 (0.36) VCAM1CASP3CASP7NPBWR1MCHR1
SCHEMBL2768514 1.00 VCAM1 (0.36) VCAM1CASP3CASP7NPBWR1MCHR1
SCHEMBL6139039 0.90 CASP3 (0.35) VCAM1CASP3CASP7NPBWR1MCHR1
SCHEMBL2768975 0.90 CASP3 (0.35) VCAM1CASP3CASP7NPBWR1MCHR1
SCHEMBL2769590 0.90 CASP3 (0.35) VCAM1CASP3CASP7NPBWR1MCHR1
SCHEMBL6138091 0.84 HDAC8 (0.37) CASP3CASP7HDAC8HDAC6HDAC1
SCHEMBL2767458 0.84 HDAC8 (0.37) CASP3CASP7HDAC8HDAC6HDAC1
SCHEMBL6564147 0.84 CASP3 (0.45) CASP3CASP7CASP9KMT2AALDH1A1
SCHEMBL2769019 0.84 HDAC8 (0.37) CASP3CASP7HDAC8HDAC6HDAC1
SCHEMBL2768886 0.76 ALDH1A1 (0.41) KMT2AALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1272175-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2005-08-31 EP disclosed
EP-1272175-A2 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2003-01-08 EP disclosed
WO-2001072960-A2 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2001-10-04 WO disclosed