SCHEMBL6139946

SCHEMBL6139946

N=C1CCCCN1c1ccc(C(C(N)=O)c2ccccc2F)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 2/20 0.40
HDAC4 P56524 13/20 0.36
GAA P10253 1/20 0.35
KCNQ2 O43526 1/20 0.34
F10 P00742 1/20 0.34
HDAC3 O15379 2/20 0.33
HDAC7 Q8WUI4 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
HDAC9 Q9UKV0 2/20 0.33
HDAC5 Q9UQL6 2/20 0.33
NCOR2 Q9Y618 2/20 0.33
USP2 O75604 1/20 0.33
ESR1 P03372 1/20 0.33
MAPT P10636 1/20 0.33
NR4A1 P22736 1/20 0.33
KMT2A Q03164 1/20 0.33
PTK2B Q14289 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HDAC1 Q13547 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6140423 0.98 HIF1A (0.40) HIF1AHDAC4GAAKCNQ2HDAC3
SCHEMBL6140774 0.83 KMT2A (0.43) GAAF10USP2ESR1MAPT
SCHEMBL6139850 0.78 HIF1A (0.38) HIF1AHDAC4GAAKCNQ2HDAC3
SCHEMBL6139855 0.78 HIF1A (0.38) HIF1AHDAC4GAAKCNQ2HDAC3
SCHEMBL17968495 0.73 GAA (0.58) HDAC4GAAHDAC3HDAC7HDAC8
SCHEMBL7166322 0.73 CYP2C9 (0.53) F10USP2ESR1MAPTNR4A1
SCHEMBL5631637 0.70 CYP1A2 (0.41) GAAF10USP2ESR1MAPT
SCHEMBL5630404 0.70 F10 (0.41) F10MAPTNPSR1
SCHEMBL28177937 0.69 SIGMAR1 (0.54) KMT2A
SCHEMBL6139947 0.68 RAB9A (0.54) MAPTNR4A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1499591-A1 CARBOXYLIC ACID AMIDES MERCK PATENT GmbH (DE) 2005-01-26 EP claimed
WO-2003093235-A1 CARBOXYLIC ACID AMIDES MERCK PATENT GMBH (DE) 2003-11-13 WO claimed