SCHEMBL6140774

SCHEMBL6140774

N=C1CCCN1c1ccc(C(C(N)=O)c2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.43
MEN1 O00255 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
HTT P42858 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.39
USP2 O75604 1/20 0.39
ESR1 P03372 1/20 0.39
MAPT P10636 1/20 0.39
NR4A1 P22736 1/20 0.39
PTK2B Q14289 1/20 0.39
ALDH1A1 P00352 1/20 0.39
F10 P00742 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 2/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6140423 0.85 HIF1A (0.40) KMT2AMEN1NPSR1HTTCYP1A2
SCHEMBL6139946 0.83 HIF1A (0.40) KMT2ANPSR1USP2ESR1MAPT
SCHEMBL6140492 0.82 MEN1 (0.40) KMT2AMEN1NPSR1HTTCYP1A2
SCHEMBL7166322 0.81 CYP2C9 (0.53) KMT2ANPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL7538698 0.75 SIGMAR1 (0.56) KMT2AMEN1CYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL6771290 0.73 ALDH1A1 (0.65) KMT2AMEN1HTTCYP1A2CYP2D6
SCHEMBL741751 0.72 MEN1 (0.58) KMT2AMEN1NPSR1CYP1A2CYP2D6
SCHEMBL1675928 0.71 CA2 (0.43) USP2MAPTALDH1A1LMNA
SCHEMBL3864473 0.70 ALDH1A1 (0.45) KMT2AMEN1NPSR1HTTUSP2
Hydrochloric Acid SCHEMBL8550499 0.70 MEN1 (0.56) KMT2AMEN1NPSR1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1499591-A1 CARBOXYLIC ACID AMIDES MERCK PATENT GmbH (DE) 2005-01-26 EP disclosed
WO-2003093235-A1 CARBOXYLIC ACID AMIDES MERCK PATENT GMBH (DE) 2003-11-13 WO disclosed