SCHEMBL6151502

SCHEMBL6151502

[CH2]/C=C/c1ccc(OC)c(OC)c1OC

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 7/20 0.59
CYP1B1 Q16678 7/20 0.59
CYP19A1 P11511 1/20 0.57
ABCG2 Q9UNQ0 1/20 0.56
CYP1A2 P05177 6/20 0.49
CYP2D6 P10635 2/20 0.49
MAPT P10636 2/20 0.49
ALDH1A1 P00352 2/20 0.49
KMT2A Q03164 2/20 0.49
POLB P06746 1/20 0.49
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
KDM4E B2RXH2 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
CHRNA7 P36544 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1045609 0.82 NFE2L2 (0.64) CYP1A1CYP1B1CYP19A1CYP1A2CYP2D6
SCHEMBL1045608 0.82 NFE2L2 (0.64) CYP1A1CYP1B1CYP19A1CYP1A2CYP2D6
SCHEMBL7862304 0.82 CYP1A1 (0.61) CYP1A1CYP1B1CYP19A1ABCG2CYP1A2
SCHEMBL14518617 0.82 CYP1A1 (0.61) CYP1A1CYP1B1CYP19A1ABCG2CYP1A2
SCHEMBL8502492 0.81 CYP1A1 (0.56) CYP1A1CYP1B1CYP19A1ABCG2CYP1A2
SCHEMBL8502491 0.81 CYP1A1 (0.56) CYP1A1CYP1B1CYP19A1ABCG2CYP1A2
SCHEMBL1480652 0.79 CYP1A1 (0.53) CYP1A1CYP1B1CYP19A1ABCG2CYP1A2
SCHEMBL8910888 0.79 CYP1A1 (0.56) CYP1A1CYP1B1CYP19A1ABCG2CYP1A2
SCHEMBL5182341 0.78 NFE2L2 (0.69) CYP1A1CYP1B1CYP19A1ABCG2CYP1A2
SCHEMBL746936 0.77 ABCG2 (0.57) CYP1A1CYP1B1CYP19A1ABCG2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6656510-B2 Antidepressants INDENA S.P.A. (IT) 2003-12-02 US claimed
US-20010020040-A1 Hyperforin derivatives, use thereof and formulations containing them INDENA S.P.A. (IT) 2001-09-06 US claimed
EP-1086071-A1 HYPERFORIN DERIVATIVES, THE USE THEREOF AND FORMULATIONS CONTAINING THEM INDENA S.p.A. (IT) 2001-03-28 EP claimed
WO-1999064388-A1 HYPERFORIN DERIVATIVES, THE USE THEREOF AND FORMULATIONS CONTAINING THEM INDENA S.P.A. (IT) 1999-12-16 WO claimed
JP-57032255-A None JP disclosed
EP-1607099-A1 Use of hyperforin derivatives as an antidepressant agent INDENA S.p.A. (IT) 2005-12-21 EP disclosed
US-6656510-B2 Antidepressants INDENA S.P.A. (IT) 2003-12-02 US disclosed
US-20010020040-A1 Hyperforin derivatives, use thereof and formulations containing them INDENA S.P.A. (IT) 2001-09-06 US disclosed
EP-1086071-A1 HYPERFORIN DERIVATIVES, THE USE THEREOF AND FORMULATIONS CONTAINING THEM INDENA S.p.A. (IT) 2001-03-28 EP disclosed
WO-1999064388-A1 HYPERFORIN DERIVATIVES, THE USE THEREOF AND FORMULATIONS CONTAINING THEM INDENA S.P.A. (IT) 1999-12-16 WO disclosed
JP-S5732255-A TRIMETHOXYPHENYL DERIVATIVE KOWA CO 1982-02-20 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010020040-A1 Hyperforin derivatives, use thereof and formulations containing them CRH, FOS, VIP CYP1A1 552/4885CYP1B1 245/4885CYP19A1 622/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.