SCHEMBL6151752

SCHEMBL6151752

Cc1cc(C)cc(C(=O)NN)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.56
ALDH1A1 P00352 4/20 0.56
MAPT P10636 4/20 0.56
GAA P10253 3/20 0.56
BLM P54132 2/20 0.56
POLB P06746 2/20 0.56
LMNA P02545 2/20 0.56
L3MBTL1 Q9Y468 2/20 0.56
NSD2 O96028 1/20 0.56
ALPL P05186 1/20 0.56
ALPI P09923 1/20 0.56
ALPG P10696 1/20 0.56
APEX1 P27695 1/20 0.56
HTT P42858 1/20 0.56
RECQL P46063 1/20 0.56
CASP6 P55212 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
TPMT P51580 1/20 0.52
HDAC3 O15379 2/20 0.47
HDAC4 P56524 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31148957 0.95 KDM4E (0.56) KDM4EALDH1A1MAPTGAABLM
SCHEMBL838851 0.87 KDM4E (0.48) KDM4EALDH1A1MAPTGAABLM
SCHEMBL1893743 0.82 KDM4E (0.68) KDM4EALDH1A1MAPTGAABLM
SCHEMBL12355763 0.81 KDM4E (0.56) KDM4EALDH1A1MAPTGAABLM
SCHEMBL8432669 0.79 POLB (0.62) KDM4EMAPTGAAPOLBLMNA
SCHEMBL661545 0.79 HDAC8 (0.69) KDM4EALDH1A1MAPTPOLBHDAC8
SCHEMBL15872015 0.78 HDAC6 (0.63) GAAPOLBTPMTHDAC3HDAC4
SCHEMBL1003295 0.78 TPMT (0.54) KDM4EALDH1A1MAPTGAAPOLB
SCHEMBL7787094 0.78 KDM4E (0.58) KDM4EALDH1A1MAPTGAABLM
SCHEMBL11341058 0.78 KDM4E (0.58) KDM4EALDH1A1MAPTGAABLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 74 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3698699-B2 2005-09-21 JP claimed
CN-1161325-C Diacyl hydrazide compounds as insecticide, intermediate for preparing said compounds and their preparing process 江苏省农药研究所 2004-08-11 CN claimed
US-20040106724-A1 Natural rubber produced from latex and composition comprising the same BRIDGESTONE CORPORATION (JP) 2004-06-03 US claimed
JP-2004514009-A 2004-05-13 JP claimed
EP-1332161-A2 DRYING PROCESSES FOR NATURAL RUBBER, STABILIZED NR COMPOSITIONS Bridgestone Corporation (JP) 2003-08-06 EP claimed
US-6531527-B2 Liquid dilution after coagulation BRIDGESTONE CORPORATION (JP) 2003-03-11 US claimed
WO-2002038667-A2 NATURAL RUBBER PRODUCED FROM LATEX AND COMPOSITION COMPRISING THE SAME BRIDGESTONE CORPORATION (JP) 2002-05-16 WO claimed
US-20020035195-A1 Viscosity-stabilizer-containing natural rubber latex and natural rubber and a production process thereof BRIDGESTONE CORPORATION 2002-03-21 US claimed
WO-2023161296-A1 CONJUGATION METHOD INVOLVING A TRANSGLUTAMINASE AT THE FC REGION COMPRISING A TRIMMED N-GLYCAN ADC THERAPEUTICS SA (CH) 2023-08-31 WO disclosed
US-11634391-B2 Compounds which are inhibitors of Notum UCL BUSINESS LTD (GB) 2023-04-25 US disclosed
EP-3843844-A1 COMPOUNDS UCL Business Ltd (GB) 2021-07-07 EP disclosed
US-20210171475-A1 COMPOUNDS UCL BUSINESS LTD (GB) 2021-06-10 US disclosed
WO-2020043866-A1 COMPOUNDS UCL BUSINESS LTD (GB) 2020-03-05 WO disclosed
EP-2906553-B1 OREXIN RECEPTOR ANTAGONISTS WHICH ARE [ORTHO BI (HETERO )ARYL]-[2-(META BI (HETERO)ARYL)-PYRROLIDIN-1-YL]-METHANONE DERIVATIVES IDORSIA PHARMACEUTICALS LTD (CH) 2019-06-26 EP disclosed
EP-0636608-A1 Derivatives of 1-benzenesulfonyl-1,3-dihydro-indol-2-one, their preparation and pharmaceutical compositions containing them SANOFI (FR) 1995-02-01 EP disclosed
EP-0636609-A1 1-Benzyl-1,3-dihydro-indol-2-one derivatives, their preparation, the pharmaceutical compositions containing them SANOFI (FR) 1995-02-01 EP disclosed
EP-0613924-A1 Natural rubber treated with viscosity stabilizers and production thereof BRIDGESTONE CORPORATION (JP) 1994-09-07 EP disclosed
EP-0581939-A1 N-SULPHONYL-2-OXOINDOLE DERIVATIVES HAVING AFFINITY FOR VASOPRESSIN AND/OR OCYTOCIN RECEPTORS SANOFI (FR) 1994-02-09 EP disclosed
WO-1993015051-A1 N-SULPHONYL-2-OXOINDOLE DERIVATIVES HAVING AFFINITY FOR VASOPRESSIN AND/OR OCYTOCIN RECEPTORS ELF SANOFI (FR) 1993-08-05 WO disclosed
US-4212867-A FOR AGRICULTURAL USE PHILAGRO (FR) 1980-07-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11634391-B2 Compounds which are inhibitors of Notum NOTUM, GOT2, GOT1 KDM4E 3907/4885ALDH1A1 1260/4885MAPT 1431/4885
US-20210171475-A1 COMPOUNDS GOT2, GOT1, OAT KDM4E 4149/4885ALDH1A1 658/4885MAPT 315/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.