SCHEMBL6152352

SCHEMBL6152352

CCCCC(c1ccc(OC(=O)C(F)(F)F)cc1)N(C(=O)CCc1ccccc1)c1ccc(OCCN2CCCC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.45
LTA4H P09960 4/20 0.42
EPHX2 P34913 1/20 0.41
HTT P42858 1/20 0.41
ESR2 Q92731 1/20 0.41
KDM4E B2RXH2 2/20 0.40
PSMB1 P20618 1/20 0.40
PSMB5 P28074 1/20 0.40
PSMB2 P49721 1/20 0.40
HRH3 Q9Y5N1 3/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5864089 0.93 EPHX2 (0.43) ESR1LTA4HEPHX2HTTESR2
SCHEMBL5863697 0.91 HTT (0.47) ESR1LTA4HEPHX2HTTESR2
SCHEMBL5863871 0.83 LTA4H (0.39) ESR1LTA4HEPHX2HTTKDM4E
SCHEMBL5864009 0.69 MMP1 (0.51) LTA4HHTTHRH3LMNAKCNH2
SCHEMBL5864176 0.68 LTA4H (0.58) ESR1LTA4HEPHX2HTTESR2
Iodobenzene SCHEMBL8059216 0.64 FAAH (0.48) LTA4H
SCHEMBL5863941 0.64 HTT (0.49) ESR1LTA4HEPHX2HTTESR2
SCHEMBL876980 0.64 LTA4H (0.75) LTA4HPSMB1PSMB5PSMB2HRH3
SCHEMBL5943719 0.64 LTA4H (0.83) LTA4HHTTPSMB1PSMB5PSMB2
SCHEMBL7134882 0.64 LTA4H (1.00) LTA4HHTTPSMB1PSMB5PSMB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542967-A1 AMIDE AND SULFONAMIDE LIGANDS FOR THE ESTROGEN RECEPTOR Pfizer Products Inc. (US) 2005-06-22 EP disclosed
WO-2004026823-A1 AMIDE AND SULFONAMIDE LIGANDS FOR THE ESTROGEN RECEPTOR PFIZER PRODUCTS INC. (US) 2004-04-01 WO disclosed