SCHEMBL6152762

SCHEMBL6152762

Cc1cc(-c2cccc(-c3ccc(OCc4ccccc4)c4c3C3CCC4C3)n2)c(C)[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.46
NOS1 P29475 1/20 0.46
NOS2 P35228 1/20 0.46
HTR1A P08908 2/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 2/20 0.38
PTGER1 P34995 1/20 0.36
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
STAT3 P40763 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KDM1A O60341 4/20 0.35
BRD4 O60885 1/20 0.35
PRMT5 O14744 4/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6153077 0.85 NOS3 (0.46) NOS3NOS1NOS2
SCHEMBL6152658 0.83 NOS3 (0.68) NOS3NOS1NOS2SMN1; SMN2CCNT1
SCHEMBL5833350 0.82 PTGER1 (0.42) NOS3NOS1NOS2PTGER1MAPT
SCHEMBL6155624 0.80 NOS3 (0.43) NOS3NOS1NOS2
SCHEMBL5834000 0.80 NOS3 (0.45) NOS3NOS1NOS2PTGER1MAPT
SCHEMBL6152763 0.80 NOS3 (0.48) NOS3NOS1NOS2HTR1ASLC6A2
SCHEMBL5834031 0.69 NOS3 (0.47) NOS3NOS1NOS2SMN1; SMN2
SCHEMBL6152928 0.68 KDM1A (0.47) HTR1ASLC6A2SLC6A4SLC6A3MAPT
SCHEMBL6700238 0.66 DRD2 (0.53)
SCHEMBL6152462 0.66 LIPE (0.55) HTR1ASLC6A2SLC6A4SLC6A3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1084109-B1 2-AMINOPYRIDINES CONTAINING FUSED RING SUBSTITUENTS AS NITRIC OXIDE SYNTHASE INHIBITORS PFIZER PROD INC (US) 2005-01-26 EP disclosed
EP-1084109-A1 2-AMINOPYRIDINES CONTAINING FUSED RING SUBSTITUENTS AS NITRIC OXIDE SYNTHASE INHIBITORS Pfizer Products Inc. (US) 2001-03-21 EP disclosed
WO-1999062883-A1 2-AMINOPYRIDINES CONTAINING FUSED RING SUBSTITUENTS AS NITRIC OXIDE SYNTHASE INHIBITORS PFIZER PRODUCTS INC. (US) 1999-12-09 WO disclosed