SCHEMBL6152658

SCHEMBL6152658

Cc1cc(-c2cccc(-c3ccc(OCCN(C)C)c4c3C3CCC4C3)n2)c(C)[nH]1

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 8/20 0.68
NOS1 P29475 8/20 0.68
NOS2 P35228 6/20 0.68
CCNT1 O60563 1/20 0.36
CDK9 P50750 1/20 0.36
HTR7 P34969 5/20 0.35
HTR1B P28222 1/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PTPN1 P18031 1/20 0.31
ROCK2 O75116 1/20 0.31
KIT P10721 1/20 0.31
KDR P35968 1/20 0.31
FLT3 P36888 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6152762 0.83 NOS3 (0.46) NOS3NOS1NOS2CCNT1CDK9
SCHEMBL6153077 0.82 NOS3 (0.46) NOS3NOS1NOS2KDM4E
SCHEMBL6583124 0.82 NOS1 (0.48) NOS3NOS1NOS2HTR7HTR1B
SCHEMBL5838088 0.81 NOS1 (1.00) NOS3NOS1NOS2
SCHEMBL5833803 0.81 NOS3 (0.67) NOS3NOS1NOS2CCNT1CDK9
SCHEMBL6152396 0.80 NOS3 (0.43) NOS3NOS1NOS2KDM4EALDH1A1
SCHEMBL6152661 0.80 NOS3 (0.71) NOS3NOS1NOS2CCNT1CDK9
SCHEMBL6155624 0.79 NOS3 (0.43) NOS3NOS1NOS2
SCHEMBL7450787 0.78 NOS3 (0.71) NOS3NOS1NOS2HTR7HTR1B
SCHEMBL6152641 0.78 NOS3 (0.38) NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1084109-B1 2-AMINOPYRIDINES CONTAINING FUSED RING SUBSTITUENTS AS NITRIC OXIDE SYNTHASE INHIBITORS PFIZER PROD INC (US) 2005-01-26 EP disclosed