SCHEMBL6153199

SCHEMBL6153199

NC(=O)N1CCCCC1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.46
GAA P10253 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
ROCK2 O75116 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
RIPK1 Q13546 1/20 0.43
KCNH2 Q12809 3/20 0.42
MCHR1 Q99705 1/20 0.42
DPP4 P27487 2/20 0.41
TACR1 P25103 1/20 0.41
HRH3 Q9Y5N1 2/20 0.41
FAP Q12884 1/20 0.41
DPP8 Q6V1X1 1/20 0.41
DPP9 Q86TI2 1/20 0.41
DPP7 Q9UHL4 1/20 0.41
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30964008 0.86 SPHK2 (0.43) OPRD1ROCK2RIPK1PDE2A
SCHEMBL5197715 0.84 CCNC (0.53) KMT2ARIPK1CCNCCDK8ALDH1A1
SCHEMBL28148131 0.84 TACR1 (0.49) OPRD1ROCK2RIPK1KCNH2MCHR1
SCHEMBL17142310 0.82 RIPK1 (0.51) OPRD1ROCK2RIPK1KCNH2MCHR1
SCHEMBL26676726 0.82 EPHX2 (0.52) GAARIPK1HRH3KDM4EALDH1A1
Trifluoroacetic Acid SCHEMBL28142751 0.82 RIPK1 (0.55) RIPK1
SCHEMBL17454889 0.81 RIPK1 (0.50) ROCK2RIPK1KCNH2MCHR1DPP4
SCHEMBL29356757 0.81 TRPC3 (0.48) GAAROCK2HPGDRIPK1ALDH1A1
SCHEMBL938757 0.80 RIPK1 (0.59) RIPK1
Trifluoroacetic Acid SCHEMBL18050102 0.77 RIPK1 (0.59) TDP1RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569646-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2005-09-07 EP disclosed
WO-2004054974-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2004-07-01 WO disclosed