SCHEMBL6156963

SCHEMBL6156963

Cc1c(O[Si](c2ccccc2)(c2ccccc2)C(C)(C)C)ccc2c(N3CCN(C)CC3)cc(=O)oc12

nearest known ligand 0.45

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.45
PDE3A Q14432 2/20 0.45
PRKDC P78527 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6156007 0.80 HSP90AA1 (0.45)
SCHEMBL6158795 0.75 HPGD (0.42)
SCHEMBL6155934 0.72 MAOB (0.43)
SCHEMBL6155892 0.71 MAOB (0.58) PRKDC
SCHEMBL5347182 0.68 PDE3B (0.66) PDE3BPDE3APRKDC
SCHEMBL5340254 0.65 PDE3B (0.71) PDE3BPDE3APRKDC
SCHEMBL5342355 0.65 PDE3B (0.63) PDE3BPDE3APRKDC
SCHEMBL6156411 0.65 PRKDC (0.49) PDE3BPDE3APRKDC
SCHEMBL6155495 0.64 MAOB (0.51) PDE3BPDE3APRKDC
SCHEMBL28365890 0.64 KMT2A (0.62) PDE3BPDE3APRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894805-B1 Ribose substituted aromatic derivatives, their preparation and use as medicaments AVENTIS PHARMA SA (FR) 2005-02-09 EP disclosed
US-5968939-A ANTIBIOTICS FROM AMINOOXOBENZOPYRAN COMPOUNDS HOECHST MARION ROUSSEL (FR) 1999-10-19 US disclosed
EP-0894805-A1 Ribose substituted aromatic derivatives, their preparation and use as medicaments HOECHST MARION ROUSSEL (FR) 1999-02-03 EP disclosed