SCHEMBL6157660

SCHEMBL6157660

CCOC(=O)/C(=N/O)c1ccc(Oc2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.52
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
HPGD P15428 1/20 0.51
CRHBP P24387 1/20 0.51
CRHR2 Q13324 1/20 0.51
ALDH1A1 P00352 3/20 0.48
HTT P42858 1/20 0.48
PARP10 Q53GL7 1/20 0.46
SRD5A2 P31213 3/20 0.45
MAPT P10636 2/20 0.45
LMNA P02545 1/20 0.45
THRB P10828 1/20 0.45
LTA4H P09960 1/20 0.45
ERCC5 P28715 1/20 0.44
FEN1 P39748 1/20 0.44
MAPK14 Q16539 1/20 0.44
HDAC3 O15379 1/20 0.44
PPARG P37231 1/20 0.44
PPARA Q07869 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6157109 1.00 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9AHPGDCRHBP
SCHEMBL6157465 1.00 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9AHPGDCRHBP
SCHEMBL6160483 0.83 ALDH1A1 (0.62) SMN1; SMN2NPC1RAB9AALDH1A1HTT
SCHEMBL6158228 0.83 ALDH1A1 (0.62) SMN1; SMN2NPC1RAB9AALDH1A1HTT
SCHEMBL6158223 0.83 ALDH1A1 (0.62) SMN1; SMN2NPC1RAB9AALDH1A1HTT
SCHEMBL16613214 0.83 NPC1 (0.49) SMN1; SMN2NPC1RAB9AHPGDCRHBP
SCHEMBL4739675 0.81 ALDH1A1 (0.57) SMN1; SMN2NPC1RAB9AHPGDCRHBP
SCHEMBL12732994 0.79 L3MBTL1 (0.51) SMN1; SMN2NPC1RAB9AALDH1A1MAPT
SCHEMBL12814773 0.79 L3MBTL1 (0.51) SMN1; SMN2NPC1RAB9AALDH1A1MAPT
SCHEMBL6340266 0.79 ALDH1A1 (0.54) SMN1; SMN2NPC1RAB9AHPGDCRHBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6924300-B2 Oxyiminoalkanoic acid derivatives TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-08-02 US disclosed
EP-1077957-B1 OXYIMINOALKANOIC ACID DERIVATIVES WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-08-04 EP disclosed
EP-1428531-A1 Oxyiminoalkanoic acid derivatives with hypoglycemic and hypolipidemic activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-06-16 EP disclosed
US-20030186985-A1 Oxyiminoalkanoic acid derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2003-10-02 US disclosed
US-6495581-B1 DRUG FOR TREATING DIABETES MELLITUS, HYPERLIPEMIA, IMPAIRED GLUCOSE TOLERANCE, ARTERIAL SCLEROSIS AND IMPROVING INSULIN RESISTANCE, INFLAMMATORY DISEASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-12-17 US disclosed
US-6251926-B1 OXYIMINOALKANOIC ACID DERIVATIVES HAVING HYPOGLYCEMIC EFFECT AND HYPOLIPIDEMIC EFFECT, IS USEFUL FOR TREATMENT OF DIABETES MELLITUS, HYPERLIPEMIA, IMPAIRED GLUCOSE TOLERANCE INFLAMMATORY DISEASE AND ARTERIOSCLEROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-06-26 US disclosed
EP-1077957-A1 OXYIMINOALKANOIC ACID DERIVATIVES WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY Takeda Chemical Industries, Ltd. (JP) 2001-02-28 EP disclosed
WO-1999058510-A1 OXYIMINOALKANOIC ACID DERIVATIVES WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-11-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030186985-A1 Oxyiminoalkanoic acid derivatives GPR119, IRS1, CPT1A SMN1; SMN2 3404/4885NPC1 1015/4885RAB9A 2830/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.