SCHEMBL6158680

SCHEMBL6158680

CC(=O)SC1CCC(=O)N(Cc2ccc(Oc3ccccc3)cc2)C1=O

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 4/20 0.46
HCRTR2 O43614 4/20 0.46
ALDH1A1 P00352 3/20 0.40
GFER P55789 1/20 0.40
LTA4H P09960 3/20 0.39
MT-CO2 P00403 1/20 0.39
ALOX5 P09917 1/20 0.39
PDPK1 O15530 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
PTPRF P10586 1/20 0.38
PTPN2 P17706 1/20 0.38
PTPN1 P18031 1/20 0.38
PTPRB P23467 1/20 0.38
ACP1 P24666 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
FAAH O00519 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6158749 0.90 HTT (0.37) HCRTR1HCRTR2HRH3
SCHEMBL6158601 0.89 ALDH1A1 (0.48) HCRTR1HCRTR2ALDH1A1MT-CO2ALOX5
SCHEMBL6157396 0.88 HCRTR1 (0.43) HCRTR1HCRTR2ALDH1A1GFERLTA4H
SCHEMBL6157016 0.82 HRH3 (0.44) HCRTR1HCRTR2LTA4HHRH3FAAH
SCHEMBL6160163 0.80 HRH3 (0.45) HCRTR1HCRTR2ALDH1A1LTA4HHRH3
SCHEMBL6160000 0.78 MEN1 (0.42) LTA4HPTGDR2PTPRFPTPN2PTPN1
SCHEMBL6157862 0.78 HCRTR1 (0.46) HCRTR1HCRTR2ALDH1A1LTA4HFAAH
SCHEMBL6159751 0.77 HCRTR1 (0.52) HCRTR1HCRTR2ALDH1A1GFERLTA4H
SCHEMBL6160031 0.77 HCRTR1 (0.49) HCRTR1HCRTR2ALDH1A1GFERLTA4H
SCHEMBL6159504 0.77 HCRTR1 (0.49) HCRTR1HCRTR2ALDH1A1GFERLTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953789-B2 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-10-11 US disclosed
US-20040157894-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-08-12 US disclosed
US-6699881-B2 MATRIX METALLOPROTEASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-03-02 US disclosed
US-20030078253-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY, LIMITED (JP) 2003-04-24 US disclosed
US-6420415-B1 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-1132379-A1 NOVEL THIOL DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND UTILIZATION THEREOF Takeda Chemical Industries, Ltd. (JP) 2001-09-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078253-A1 Thiol compounds, their production and use TST, QSOX1, SULT1E1 HCRTR1 1949/4885HCRTR2 1842/4885ALDH1A1 905/4885
US-20040157894-A1 Thiol compounds, their production and use TST, SULT1E1, QSOX1 HCRTR1 1930/4885HCRTR2 1754/4885ALDH1A1 877/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.