SCHEMBL6160163

SCHEMBL6160163

CC(=O)SC1CCCN(Cc2ccc(Oc3ccccc3)cc2)C1=O

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.45
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
EGLN1 Q9GZT9 1/20 0.41
SRC P12931 3/20 0.41
FFAR1 O14842 1/20 0.41
LTA4H P09960 5/20 0.41
HCRTR1 O43613 2/20 0.40
HCRTR2 O43614 2/20 0.40
MMP8 P22894 1/20 0.40
MMP12 P39900 1/20 0.40
MMP13 P45452 1/20 0.40
FAAH O00519 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6157016 0.93 HRH3 (0.44) HRH3EGLN1LTA4HHCRTR1HCRTR2
SCHEMBL6158696 0.88 SRC (0.45) HRH3EGLN1SRCFFAR1LTA4H
SCHEMBL6159709 0.81 LTA4H (0.44) HRH3EGLN1SRCLTA4HFAAH
SCHEMBL6158680 0.80 HCRTR1 (0.46) HRH3ALDH1A1LTA4HHCRTR1HCRTR2
SCHEMBL6159308 0.80 HRH3 (0.48) HRH3EGLN1SRCFFAR1LTA4H
SCHEMBL6158267 0.78 HRH3 (0.49) HRH3EGLN1SRCFFAR1LTA4H
SCHEMBL6159991 0.78 HRH3 (0.42) HRH3ALDH1A1EGLN1LTA4HHCRTR1
SCHEMBL6158601 0.77 ALDH1A1 (0.48) ALDH1A1HCRTR1HCRTR2
SCHEMBL6158966 0.76 MEN1 (0.43) HRH3EGLN1LTA4HHCRTR1HCRTR2
SCHEMBL6158954 0.76 MEN1 (0.43) HRH3EGLN1LTA4HHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953789-B2 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-10-11 US disclosed
US-20040157894-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-08-12 US disclosed
US-6699881-B2 MATRIX METALLOPROTEASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-03-02 US disclosed
US-20030078253-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY, LIMITED (JP) 2003-04-24 US disclosed
US-6420415-B1 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-1132379-A1 NOVEL THIOL DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND UTILIZATION THEREOF Takeda Chemical Industries, Ltd. (JP) 2001-09-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078253-A1 Thiol compounds, their production and use TST, QSOX1, SULT1E1 HRH3 505/4885ALDH1A1 905/4885MAPK1 2637/4885
US-20040157894-A1 Thiol compounds, their production and use TST, SULT1E1, QSOX1 HRH3 463/4885ALDH1A1 877/4885MAPK1 2685/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.